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Estrenes

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Definition: Unsaturated derivatives of the ESTRANES with methyl groups at carbon-13, with no carbon at carbon-10, and with no more than one carbon at carbon-17. They must contain one or more double bonds.  do not confuse with ESTRANES   
Examples Allylestrenol; Epimestrol; Equilenin; Equilin; Estradiol; Estriol; Estrone; Metribolone; Mifepristone; Nandrolone; Trenbolone Acetate 		Other names 19-Norandrostenes; 19 Norandrostenes
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
17-beta-O-(1-(2-carboxy-(2-hydroxy-4-methoxy-3-carboxamido)anilido)ethyl)1,3,5(10)-estratriene  0   *Estrenes. Bioorg Med Chem Lett. 2010 Dec 15;20(24):7450-3
11-(4-(N-methyl-N-cyclohexylmethylamino)phenyl)-17-(1-propinyl)-17-hydroxyl-4,9-estradiene-3-one  0   *Estrenes. J Chromatogr B Analyt Technol Biomed Life Sci 2010 Mar;878(7-8):719-23
(6-(2-aminoethylamino)hexyl)carbamic acid 2-(6-(7-estra-1,3,5,(10)-triene)hexylamino)ethyl ester platinum(II) dichloride  0   *Estrenes *Organoplatinum Compounds. J Inorg Biochem 2009 Feb;103(2):256-61
2-methoxyoestra-1,3,5(10),16-tetraene-3-carboxamide  0   *Estrenes. Anticancer Res 2008 May-Jun;28(3A):1483-91
2-methoxyestradiol-3,17-O,O-bis(sulfamate)  0   *Estrenes. Br J Cancer 2007 Dec 17;97(12):1673-82
2-methoxy-3-O-sulfamoyl-17-cyanomethylestra-1,3,5(10)-triene  0   *Estrenes. Br J Cancer 2007 Dec 17;97(12):1673-82
17beta-acetoxy-2-fluoro-3-methoxy-8alpha-estra-1,3,5(10)-triene  0   *Estrenes. Bioorg Khim. 2007 May-Jun;33(3):315-23
10beta-chloro-17beta-hydroxyestra-1,4-dien-3-one  0   *Estrenes. Steroids. 2006 Aug;71(8):670-3
asoprisnil  0 benzaldehyde, 4-((11beta, 17beta)-17-methoxy-17-(methoxymethyl)-3-oxoestra-4, 9-dien-11beta-yl)-, 1-oxime  *Estrenes *Oximes Oxytocics. Steroids. 2003 Nov;68(10-13):1019-32
4-estren-3,17-diol  0   *Estrenes. Science.2002 Oct 25;298(5594):843-6
puboestrene  0   *Estrenes. Phytochemistry 2001 Dec;58(8):1199-204
4-(17beta-methoxy-17alpha-(methoymethyl)-3-oxoestra-4,9-dien-11beta-yl)benzaldehyd-1-(E)-(O-(ethylamino)carbonyl)oxime  0   *Estrenes *Oximes Oxytocics. J Reprod Fertil Suppl 2001;57():249-54
ZK 230211  0   *Estrenes Receptors, Progesterone/antagonists & inhibitors. J Med Chem 2000 Dec 28;43(26):5010-6
aglepristone  124478-60-0   *Estrenes. Schweiz Arch Tierheilkd. 2000 Jul;142(7) :381-6
4-(17-methoxy-17-(methoxymethyl)-estra-4,9-dien-11-yl)benzaldehyd-1-oxime  0   *Estrenes. Pharmazie 2000 Jun;55(6):463-4
17-hydroxy-11-(3'-sulfanylpropyl)oxy-estra-1,3,5(10)-trien-3-yl sulfamate  0   *Estrenes *Sulfonic Acids Haptens. Steroids 1999 Jul;64(7):460-71
RTI 3021-022  0   *Estrenes. Endocrinology 1999 Mar;140(3):1449-58
RTI 3021-012  0   *Estrenes. Endocrinology 1999 Mar;140(3):1449-58
3-(n-dimethylaminoethyloxy)estra-1,3,5-triene  0   *Estrenes. J Steroid Biochem Mol Biol 1996 Sep;59(1):49-54
3-methoxy-14,15-methylenestra-1,3,5(10),8-tetraen-17-ol  0   *Estrenes. Steroids 1996 Feb;61(2):48-9
10-(1-azirinyl)estr-4-en-3,17-dione  0   *Estrenes. Steroids 1996 Mar;61(3):138-43
Org 20781  0   *Estrenes. J Pharm Pharmacol 1995 Jul;47(7):608-13
EM 219  0   *Estrenes. Breast Cancer Res Treat 1995 May;34(2):147-59
Org 33628  0   *Estrenes. Ann N Y Acad Sci 1995 Jun 12;761:192-201
pentolame  150748-24-6 17-beta-(5-hydroxy-1-pentylamino)-1,3,5(10)-estratrien-3-ol  *Amino Alcohols *Estrenes Estradiol Congeners. Proc West Pharmacol Soc 1993;36:143-7
butolame  150748-23-5 17 beta-(4-hydroxy-1-butylamino)-1,3,5(10)-estratrien-3-ol  *Amino Alcohols *Estrenes. Proc West Pharmacol Soc 1993;36:143-7
4-(3-hydroxyestra-1,3,5(10)-tetraen-16-yl)-2-methylene-4-butanolide  150585-14-1   *Estrenes 4-Butyrolactone/*analogs & derivatives. Steroids 1993 May;58(5):234-8
estra-1,3,5(10)-trien-17-one-3-sulfonyl chloride  148259-10-3   *Estrenes *Sulfones. Steroids 1993 Mar;58(3):106-11
3,3,17,17-bis(ethylenedioxy)-5,10-oxidoestr-9(11)-ene  55180-24-0   *Estrenes. Steroids 1992 Apr;57(4):154-61
3-hydroxyestra-1,3,5(10),6-tetraen-17-one  2208-12-0   *Estrenes. Biochemistry 1992 Aug 25;31(33):7609-21
Org 31806  123916-70-1   *Estrenes *Furans. J Steroid Biochem Mol Biol 1992 Aug;42(7):695-704
Org 31710  118968-41-5   *Estrenes *Furans. J Steroid Biochem Mol Biol 1992 Aug;42(7):695-704
U 73343  142878-12-4   *Estrenes *Pyrrolidinones Type C Phospholipases/antagonists & inhibitors. Endocrinology 1992 Jun;130(6):3475-83
10-methylthioethyl estra-4,9(11)-diene 3,17-dione  137437-16-2 Estra-4,9(11)-diene-3,17-dione, 10-(2-(methylthio)ethyl)  *Estrenes Aromatase Inhibitors. J Steroid Biochem Mol Biol 1992 Mar;41(3-8):773-7
methylestrenolone  514-61-4 estr-4-en-3-one, 17-beta-hydroxy-17-alpha-methyl  *Estrenes Progesterone Congeners.
N-chloro-3-methoxy-16-aza-1,3,5(10)-estratrien-17-one  114462-28-1   *Azasteroids *Estrenes. Acta Crystallogr B 1991;47(Pt 3):383
N-chloro-3-methoxy-17-aza-homo-1,3,5(10)-estratrien-17-one  114462-29-2   *Azasteroids *Estrenes. Acta Crystallogr B 1991;47(Pt 3):383
N-chloro-3-methoxy-17-azahomo-1,3,5(10)-estratrien-16-one  119111-52-3   *Azasteroids *Estrenes. Acta Crystallogr B 1991;47(Pt 3):383
trendione  4642-95-9   *Estrenes. J Chromatogr 1991;564(2):485
pyridinium 3-methoxyestra-1,3,5(10)-trien-6-yl sulfate  134223-97-5   *Estrenes *Pyridinium Compounds. Steroids 1991;56(4):173
6,6'-bi(7-allyl-3-oxo-4-estren-17-yl acetate)  119020-36-9   *Allyl Compounds *Estrenes. Acta Crystallogr C 1991;47(Pt 3):689
17-(N,N-diisopropylcarbamoyl)estra-1,3,5(10)-triene-3-sulfonic acid  131267-92-0   *Estrenes 3-Oxo-5-alpha-Steroid 4-Dehydrogenase/antagonists & inhibitors. Steroids 1991;56(1):4
17-(N-t-butylcarboxamide)estra-1,3,5(10)-triene-3-carboxylic acid  124651-01-0   *Estrenes 3-Oxo-5-alpha-Steroid 4-Dehydrogenase/antagonists & inhibitors. J Steroid Biochem Mol Biol 1990;37(4):575
17-(N,N-diisopropylcarboxamide)estra-1,3,5(10)-triene-3-carboxylic acid  124650-99-3   *Estrenes 3-Oxo-5-alpha-Steroid 4-Dehydrogenase/antagonists & inhibitors. J Steroid Biochem Mol Biol 1990;37(4):575
benz(3,4)-6-oxaestra-1,3,5(10),8-tetraen-17-ol  131077-42-4   *Estrenes *Steroids, Heterocyclic. Steroids 1990;553):101
hexolame  110346-23-1 Estra-1,3,5(10)-trien-3-ol, 17-((6-hydroxyhexyl)amino)-, (17beta)  *Amino Alcohols *Estrenes Estradiol Congeners. Steroids 1990;55(2):83
17-hydroxy-7-methyl-D-homoestra-4,16-dien-3-one  103742-75-2   *Estrenes *Homosteroids. Steroids 1990;55(2):59
17-propynylestra-1,3,5-triene-3,17-diol dicyclopentadienyl dimolybdenum tetracarbonyl  101859-58-9   *Estrenes *Organometallic Compounds Molybdenum. J Steroid Biochem 1989;34(1-6):301
17-propynylestra-1,3,4(10)-triene-3,17-diol dicobalt hexacarbonyl  101859-59-0   *Estrenes *Organometallic Compounds Cobalt. J Steroid Biochem 1989;34(1-6):301
Org 7797  80177-51-1 Estra-1,3,5(10)-triene-3,16-diol, 17-(methylamino)-, (16alpha,17beta)-, (Z)-2-butenedioate (1:1) (salt)  *Estrenes. J Cardiovasc Pharmacol 1989;14(2):205
1-(6-((3-methoxyestra-1,3,5(10)-trien-17-yl)amino)hexyl)-1H-pyrrole-2,5-dione  112648-68-7 1H-Pyrrole-2,5-dione, 1-(6-(((17beta)-3-methoxyestra-1,3,5(10)-trien-17-yl)amino)hexyl)  *Estrenes *Pyrrolidinones Type C Phospholipases/antagonists & inhibitors.
Pharma Action Phosphodiesterase Inhibitors ; Platelet Aggregation Inhibitors 		Adv Prostaglandin Thromboxane Leukotriene Res 1989;19:590
10-chloroestradien-3-one  0   *Estrenes. J Steroid Biochem 1988;31(5):867
U 26384  112646-88-5   *Estrenes Phospholipases A/antagonists & inhibitors. J Clin Invest 1988;82(4):1333
SC 35135  90733-42-9 Estr-5-ene-3,17-dione, 10-(2-aminoethyl)-, cyclic bis(1,2-ethanediyl acetal), acetate  *Estrenes. J Cardiovasc Pharmacol 1988;12(2):218
3-hydroxy-14,15-secoestra-1,3,5(10)-trien-15-yn-17-one  117144-19-1   *Estrenes *Secosteroids Estradiol Dehydrogenases/antagonists & inhibitors. J Biol Chem 1988;263(24):11640
2,3-bisaza-A-nor-1,5(10)-estradien-17-ol  89288-70-0   *Azasteroids *Estrenes. Steroids 1986;48(3-4):213
6,7-benzo-3-methoxyestra-1,3,5(10),8,14-pentaen-17-one  115375-36-5   *Estrenes. Steroids 1986;48(5-6):401
17 beta-hydroxy-7 alpha-methyl-5-estren-3-one  50718-35-9   *Estrenes. Exp Clin Endocrinol 1987;89(2):174
10-thiirane-4-estrene-3,17-dione  108180-16-1   *Estrenes Aromatase Inhibitors. J Biol Chem 1987;262(9):4421
10-oxirane-4-estrene-3,17-dione  108180-14-9   *Estrenes Aromatase Inhibitors. J Biol Chem 1987;262(9):4421
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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012
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