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Indium Radioisotopes

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Definition: Unstable isotopes of indium that decay or disintegrate emitting radiation. In atoms with atomic weights 106-112, 113m, 114, and 116-124 are radioactive indium isotopes.  In-106-112, 113m, 114, 116-124; /blood-csf-urine /metab permitted but not for tracer studies (    Other names Radioisotopes, Indium
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
111In-nuclear translocation sequence-7G3  0   *Antibodies, Monoclonal *Coordination Complexes Indium Radioisotopes. J Nucl Med 2011 Sep;52(9):1465-73
111In-DOTA-p-nitrophenylalanyl-cyclo(cysteinyl-tyrosyl-tryptophyl-lysyl-threonyl-cysteinyl)tyrosinamide  0   *Peptides, Cyclic *Coordination Complexes Indium Radioisotopes Receptors, Somatostatin/antagonists & inhibitors. J Nucl Med 2011 Sep;52(9):1412-7
DTPA(1)-Lys(3),Tyr(4)bombesin  0   *Pentetic Acid Bombesin/*analogs & derivatives Indium Radioisotopes. Cancer Biother Radiopharm. 2009 Aug;24(4):435-43
111In-DTPA-trastuzumab  0   *Organometallic Compounds *Antibodies, Monoclonal, Humanized Indium Radioisotopes. Eur J Nucl Med Mol Imaging 2009 Jan;36(1):81-93
111In-DOTA-cyclo(arginyl-glycyl-aspartyl-phenylalanyl-lysyl)  0   *Organometallic Compounds *Peptides, Cyclic Indium Radioisotopes. Eur J Nucl Med Mol Imaging 2008 Aug;35(8):1507-15
111In-CHX-A''-DTPA-Z(HER2;342) affibody  0   *Recombinant Fusion Proteins Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Q J Nucl Med Mol Imaging 2007 Dec;51(4):314-23
indium-111-DTPA-CTT  0   *Peptides, Cyclic Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 2007 Jul;34(5):503-10
111In-DOTA-Z(HER2-342-pep2)  0   *Organometallic Compounds *Recombinant Fusion Proteins Indium Radioisotopes. Cancer Res 2007 Mar 1;67(5):2178-86
(Lys(40)(Ahx-DTPA-111In)NH2)exendin-14  0   *Organometallic Compounds *Peptides Indium Radioisotopes. J Nucl Med 2006 Dec;47(12):2025-33
111indium-DTPA-Ac-TZ14011  0   *Peptides, Cyclic Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 2006 May;33(4):489-94
111In-benzyl-DTPA-ZHER2:342  0   *Receptor, erbB-2 Pentetic Acid/*analogs & derivatives Indium Radioisotopes. J Nucl Med. 2006 May;47(5):846-53
111In-DOTA-TOC  0   Octreotide/*analogs & derivatives Indium Radioisotopes. Eur J Nucl Med Mol Imaging 2005 Oct;32(10):1144-51
111In-diDTPA-FKYK  0   *Oligopeptides Pentetic Acid/*analogs & derivatives Indium Radioisotopes. J Nucl Med. 2005 Mar;46(3):495-501
111In-octreotate, DOTA(0)-Tyr(3)-Thr(8)  0   *Organometallic Compounds Octreotide/*analogs & derivatives Indium Radioisotopes. Eur J Nucl Med Mol Imaging 2004 Sep;31(9):1257-62
111In-octreotide, DTPA(0)  0   Pentetic Acid/*analogs & derivatives Octreotide/*analogs & derivatives Indium Radioisotopes. J Nucl Med 2005 Jan;46 Suppl 1:62S-6S
DTPA pentetreotide  0   Pentetic Acid/*analogs & derivatives Indium Radioisotopes.
Pharma Action Indicators and Reagents
J Clin Endocrinol Metab 2002 Apr;87(4):1627-33
111In-DTPA-N-TIMP-2  0   *Tissue Inhibitor of Metalloproteinase-2 Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Eur J Nucl Med 2001 Jun;28(6):756-61
In-DOTA-NSC-ST  0   *Heterocyclic Compounds, 1-Ring Indium Radioisotopes. Anticancer Res 2001 Jul-Aug;21(4A):2785-92
N,N-bis(2-(bis(n-heptylcarbamoyl)amino)ethyl)glycine  0   Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 2000 Aug;27(6):605-10
N,N-bis(2-(bis(2-ethylhexylcarbamoylethyl)amino)ethyl)glycine  0   Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 2000 Aug;27(6):605-10
DTPA-methotrexate  0   Pentetic Acid/*analogs & derivatives Methotrexate/*analogs & derivatives Indium Radioisotopes. Cancer Biother Radiopharm 1998 Jun;13(3):177-84
DOTALAN  0   *Heterocyclic Compounds, 1-Ring *Peptides, Cyclic Indium Radioisotopes Yttrium Radioisotopes. Endocrinology 1999 Nov;140(11):5136-48
DTPA-Pro(1),Tyr(4)bombesin  0   *Pentetic Acid Bombesin/*analogs & derivatives Indium Radioisotopes. Int J Cancer 1999 Nov 26;83(5):657-63
indium DTPA-adriamycin  0   Doxorubicin/*analogs & derivatives Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Anticancer Drugs 1999 Jan;10(1):89-95
111-indium-ethylenediaminetetracetic acid-biotin  0   Biotin/*analogs & derivatives Edetic Acid/*analogs & derivatives Contrast Media Indium Radioisotopes. J Nucl Med 1999 Mar;40(3):484-90
indium 111-cT84.66 monoclonal antibody  0   *Antibodies, Monoclonal *Immunoglobulin G Indium Radioisotopes. J Nucl Med 1998 Dec;39(12):2097-104
indium 111-DOTA-lanreotide  0   *Heterocyclic Compounds *Peptides, Cyclic Indium Radioisotopes. J Nucl Med 1998 Dec;39(12):2090-4
DTPA-heparin  0   Pentetic Acid/*analogs & derivatives Heparin/*analogs & derivatives Indium Radioisotopes. Thromb Res 1998 Jan 1;89(1):23-30
indium DTPA-RC-160  0   *Oligopeptides Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Eur J Nucl Med 1998 Feb;25(2):182-6
indium benzyldiethylenetriaminepentaacetic acid  0   Pentetic Acid/*analogs & derivatives Indium Radioisotopes. J Med Chem 1997 Nov 21;40(24):3986-9
DTPA folate  0   Pentetic Acid/*analogs & derivatives Folic Acid/*analogs & derivatives Indium Radioisotopes. Bioconjug Chem 1997 Sep-Oct;8(5):673-9
indium DTPA-epsilon-lysine  0   Pentetic Acid/*analogs & derivatives Lysine/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 1994 Nov;21(8):1023-34
(DOTA(0)-Phe(1)-Tyr(3))octreotide  0   Octreotide/*analogs & derivatives Indium Radioisotopes Yttrium Radioisotopes.
Pharma Action Radiopharmaceuticals
Eur J Nucl Med;1997 Apr;24(4):368-71
indium DTPA-albumin  0   *Albumins Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 1996 Jul;23(5):595-8
alpha,omega-(bis)DTPA-biocytin  0   Pentetic Acid/*analogs & derivatives Lysine/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 1996 May;23(4):459-66
Capromab Pendetide  145464-28-4   *Antibodies, Monoclonal Indium Radioisotopes Prostatic Neoplasms.
Pharma Action Indicators and Reagents
J Nucl Med;1996 Sep;37(9):1583-8PROSTASCINT
indium DTPA-bis(stearylamide)  0   *Stearates Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Bioconjug Chem 1996 Jan-Feb;7(1):72-81
substance P, Indium-111-DTPA-Arg(1)  0   Pentetic Acid/*analogs & derivatives Substance P/*analogs & derivatives Indium Radioisotopes. J Nucl Med 1996 Jan;37(1):108-17
indium polylysine-EAK  0   Polylysine/*analogs & derivatives Indium Radioisotopes. J Nucl Biol Med 1994 Dec;38(4 Suppl 1):104-8
DTPA-B2  0   Biotin/*analogs & derivatives Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Commun 1995 Jan;16(1):38-46
biotinyl-hydrazino-EDTA  0   Biotin/*analogs & derivatives Edetic Acid/*analogs & derivatives Indium Radioisotopes Organotechnetium Compounds. Nucl Med Commun 1995 Jan;16(1):38-46
indium-111-octreotide  0   Octreotide/*analogs & derivatives Indium Radioisotopes.
Pharma Action Radiopharmaceuticals
J Nucl Biol Med 1994 Dec;38(4):576-8
indium-ethylenedicysteine  0   *Organometallic Compounds Cysteine/*analogs & derivatives Indium Radioisotopes. Nucl Med Biol 1995 Feb;22(2):165-73
N-alpha-DTPA-tyrosyl-N-epsilon-DTPA-lysine  0   *Dipeptides Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Commun 1994 Dec;15(12):972-80
pentetreotide  138661-02-6 L-Cysteinamide, N-(2-((2-(bis(carboxymethyl)amino)ethyl)(carboxymethyl)amino)ethyl)-N-(carboxymethyl)glycyl-D-phenylalanyl-L-cysteinyl-L-phenylalanyl-D-tryptophyl-L-lysyl-L-threonyl-N-(2-hydroxy-1-(hydroxymethyl)propyl)-, cyclic (3-8)-disulfide, (R-,(R*,  Somatostatin/*analogs & derivatives Indium Radioisotopes. Br J Cancer 1993 Jun;67(6):1437-9OCTREOSCAN
monoclonal antibody ZCE 025  139039-70-6   *Antibodies, Monoclonal Carcinoembryonic Antigen Indium Radioisotopes. Cancer 1993 Jun 15;71(12 Suppl):4293-7
ATN 10  134837-80-2   *Deuteroporphyrins Indium Radioisotopes. Nucl Med Biol 1993 Feb;20(2):231-7
(111)In-Fab-DTPA antimyosine  0   *Immunoglobulin Fab Fragments Pentetic Acid/*analogs & derivatives Indium Radioisotopes Myosins. J Nucl Med 1993 Feb;34(2):234-41
indium In 113m sulfur colloid  0   *Indium *Sulfur Colloids Indium Radioisotopes. Nucl Med Commun 1992 Nov;13(11):817-23
SDZ 215-811  142694-57-3   Pentetic Acid/*analogs & derivatives Octreotide/*analogs & derivatives Indium Radioisotopes Terbium.
Pharma Action Radiopharmaceuticals
Life Sci 1991;49(22):1583
DTPA-IgG complex  0   *Immunoglobulin G Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Nucl Med Commun 1991;12(3):175
indium(111)-ethylenediamine-N,N'-bis(2-hydroxyphenylacetic acid)  132830-15-0   *Ethylenediamines Indium Radioisotopes. J Nucl Med 1990;31(10):1662
Indium 111In-satumomab pendetide  0   *Oligopeptides *Antibodies, Monoclonal Pentetic Acid/*analogs & derivatives Indium Radioisotopes. Radiology 1990;175(1):163MPI INDIUM DTPA IN 111
indium 1-(4-isothiocyanatobenzyl)ethylenediaminetetraacetic acid  0   *Organometallic Compounds Edetic Acid/*analogs & derivatives Indium Indium Radioisotopes. J Nucl Med 1990;31(2):218
imciromab pentetate  138660-99-8   *Antibodies, Monoclonal *Organometallic Compounds Indium Indium Radioisotopes Myosins. Rev Esp Cardiol 1988;41 Suppl 2:70MYOSCINT
indium 1-(4-isothiocyanatobenzyl)diethylenetriaminepentaacetic acid  0   *Organometallic Compounds Pentetic Acid/*analogs & derivatives Indium Indium Radioisotopes. J Nucl Med 1988;29(11):1810
ATN-2  119130-46-0   *Porphyrins Indium Radioisotopes. Jpn J Cancer Res 1988;79(7):880
indifor  124399-52-6   *Organophosphorus Compounds Indium Radioisotopes. Med Radiol (Mosk) 1986;31(7):53
indium-bleomycin  0   *Organometallic Compounds Bleomycin/*analogs & derivatives Indium Radioisotopes. J Surg Oncol 1985;29(2):71
indium ferric colloid  0   *Ferric Compounds *Indium Colloids Indium Radioisotopes. Exp Hematol 1985;13(1):1
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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012

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