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Ketanserin

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Definition: A selective serotonin receptor antagonist with weak adrenergic receptor blocking properties. The drug is effective in lowering blood pressure in essential hypertension. It also inhibits platelet aggregation. It is well tolerated and is particularly effective in older patients.     
Pharmacological Action Antihypertensive Agents; Platelet Aggregation Inhibitors; Serotonin Antagonists 		Other names R41468; R41,468; R 41468; R 41,468; R-41468; R-41,468; 3-(2-(4-(4-Fluorobenzoyl)piperidinol)ethyl)-2,4(1H
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
altanserin  76330-71-7 4(1H)-Quinazolinone, 3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)-2,3-dihydro-2-thioxo  Ketanserin/*analogs & derivatives Fluorine Radioisotopes Ligands. J Nucl Med 1991;32(12):2266
N-2-fluoroethylketanserin  136346-26-4   Ketanserin/*analogs & derivatives. Neurosci Lett 1991;123(1):23
azidoiodoketanserin  136769-36-3   Ketanserin/*analogs & derivatives *Azides Iodine Radioisotopes. Eur J Pharmacol 1990;186(1):95
6-hydroxyketanserin  94840-70-7   Ketanserin/*analogs & derivatives. Arzneimittelforschung 1988;38(6):785
Poly-5  0   *Cimetidine *Diphenhydramine *Ibuprofen *Ketanserin *Methylprednisolone Drug Combinations. J Trauma 1987;27(12):1313
7-amino-8-iodoketanserin  105554-25-4   Ketanserin/*analogs & derivatives. Biochem Pharmacol 1986;35(19):3199
7-aminoketanserin  102745-99-3   Ketanserin/*analogs & derivatives. J Med Chem 1986;29(9):1663
butanserin  87051-46-5   Ketanserin/*analogs & derivatives. J Pharm Pharmacol 1986;38(5):374
6-azidoketanserin  97930-92-2 2,4(1H,3H)-Quinazolinedione, 6-azido-3-(2-(4-(4-fluorobenzoyl)-1-piperidinyl)ethyl)  *Azides Ketanserin/*analogs & derivatives. J Biol Chem 1985;260(14):8423
7-azidoketanserin  95653-71-7   *Azides Ketanserin/*analogs & derivatives. FEBS Lett 1985;182(2):291
ketanserinol  76330-73-9 2,4(1H,3H)-Quinazolinedione, 3-(2-(4-((4-fluorophenyl)hydroxymethyl)-1-piperidinyl)ethyl)  Ketanserin/*analogs & derivatives. J Chromatogr 1983;277:396

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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012
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