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Naloxone

More information in Books or onNLM PubMed
Definition: A specific opiate antagonist that has no agonist activity. It is a competitive antagonist at mu, delta, and kappa opioid receptors.     
Pharmacological Action Narcotic Antagonists
Examples Naltrexone 		Other names Naloxonratiopharm; Naloxon ratiopharm; MRZ2593; MRZ 2593Br; MRZ 2593 Br; MRZ 2593; Hydrochloride, Naloxone; Hydrochloride Dihydride, Naloxone; Hydrobromide, Naloxone; Curamed, Naloxon; Bristol Myers Squibb Brand of Naloxone Hydrochlori; Dihydride, Naloxone Hydrochloride; Abello, Naloxone; ratiopharm Brand of Naloxone Hydrochloride; United Drug Brand of Naloxone Hydrochloride; SERB Brand of Naloxone Hydrochloride; Narcanti; Narcan; Naloxone, (5 beta,9 alpha,13 alpha,14 alpha)-Isome; Naloxone Hydrochloride, (5 beta,9 alpha,13 alpha,1Drugs* : NARCAN; NALOXONE; NALOXONE HCL; NALOXONE HYDROCHLORIDE
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
oxycodone naloxone combination  0   *Naloxone *Oxycodone Drug Combinations Constipation/prevention & control Delayed-Action Preparations. Drug Ther Bull. 2010 Dec;48(12):138-41
naloxone-3-glucuronide  0   Naloxone/*analogs & derivatives. Dig Dis Sci 2007 Feb;52(2):502-7
suboxone  0   *Buprenorphine *Naloxone Drug Combinations. Am J Addict 2006 Jan-Feb;15(1):1-7SUBOXONE
N-cubylmethylnoroxymorphone  0   Naloxone/*analogs & derivatives. Bioorg Med Chem 1996 Jan;4(1):73-80
naloxone-3-O-methyl-oxime  0   Naloxone/*analogs & derivatives. Neurochem Res 1994 Sep;19(9):1159-63
naloxone benzoylhydrazone  119630-94-3 Benzoic acid, ((5alpha)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene)hydrazide  Naloxone/*analogs & derivatives. Mol Pharmacol 1989;35(1):67
estrone-naloxone azine  91712-59-3   Estrone/*analogs & derivatives Naloxone/*analogs & derivatives. Natl Inst Drug Abuse Res Monogr Ser 1986;75:45
talwin Nx  126663-39-6   *Naloxone *Pentazocine Drug Combinations. JAMA 1986;256(18):2562PENTAZOCINE AND NALOXONE HYDROCHLORIDES; PENTAZOCINE AND NALOXONE HYDROCHLORIDE; TALWIN NX
naloxazine  71786-91-9   Naloxone/*analogs & derivatives. Yao Hsueh Hsueh Pao 1984;19(4):251
14-hydroxydihydromorphazine  97345-76-1 Morphinan-3,14-diol, 4,5-epoxy-6-hydrazino-17-methyl-, (5alpha)  Naloxone/*analogs & derivatives. Yao Hsueh Hsueh Pao 1984;19(4):251
N-methylnaloxone  73232-50-5   Quaternary Ammonium Compounds Naloxone/*analogs & derivatives. J Pharmacol Exp Ther 1984;229(2):481
naloxone-6-spirohydantoin  87872-71-7 Spiro(imidazolidine-4,6'-morphinan)-2,5-dione, 4',5'-epoxy-3',14'-dihydroxy-17'-(2-propenyl)-, (5'alpha)  *Hydantoins Naloxone/*analogs & derivatives. Neuropharmacology 1983;22(9):1151
naloxonazine  82824-01-9 Morphinan-6-one, 4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)-, ((5alpha)-4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)morphinan-6-ylidene)hydrazone, (5alpha)  Naloxone/*analogs & derivatives. J Neurosci 1982;2(5):572
Valoron N  0   *Naloxone *Tilidine Drug Combinations. ZFA (Stuttgart) 1980;56(7):505
naloxazone  73674-85-8 Morphinan-6-one, 4,5-epoxy-3,14-dihydroxy-17-(2-propenyl)-, hydrazone, (5alpha)  Naloxone/*analogs & derivatives. Science 1980; 208(4443):514
6 beta-naloxol  53154-12-4 (5 alpha,6 beta)-4,5-epoxy-17-(2-propenyl)morphinan-3,6,14-triol  Naloxone/*analogs & derivatives. Comp Biochem Physiol (C) 1980;65(2):93
6 alpha-naloxol  20410-95-1 (5 alpha,6 alpha)-4,5-epoxy-17-(2-propenyl)morphinan-3,6,14-triol  Naloxone/*analogs & derivatives. Comp Biochem Physiol (C) 1980;65(2):93
nalmexone  16676-26-9 4,5-epoxy-3,14-dihydroxy-17-(3-methyl-2-butenyl)morphinan-6-one  Naloxone/*analogs & derivatives.
naloxone-3-ethereal sulfate  34707-87-4   Naloxone/*analogs & derivatives. Proc Soc Exptl Biol Med 139(3):865;1972

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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012
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