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Receptors, Angiotensin

More information in Books or onNLM PubMed
Definition: Cell surface proteins that bind ANGIOTENSINS and trigger intracellular changes influencing the behavior of cells.  note specific subtypes; do not confuse receptors that bind to ANGIOTENSIN II and ANGIOTENSIN III with specific angiotensin receptor subtypes   
Examples Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2
Other names Angiotensin Receptors; Receptor, Angiotensin III; Receptor, Angiotensin II; Angiotensin III Receptor; Angiotensin II Receptor
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
N-butyloxycarbonyl-3-(4-(2-oxopyrrolidin-1-ylmethyl)phenyl)-5-isobutylthiophene-2-sulfonamide  0   *Sulfonamides *Thiophenes Receptors, Angiotensin/agonists. Bioorg Med Chem 2010 Jun 15;18(12):4570-90
3-(1-biphenyl-4-ylmethyl-3-ethoxycarbonyl-1-butylcarbamoyl)propionate-3'-methyl-2'-(pentanoyl(2'-(tetrazol-5-ylate)biphenyl-4'-ylmethyl)amino)butyrate  0   *Aminobutyric Acids *Tetrazoles Receptors, Angiotensin/antagonists & inhibitors Neprilysin/antagonists & inhibitors. Lancet 2010 Apr 10;375(9722):1255-66
Agtrap protein, rat  0   *Receptors, Angiotensin. Hypertension 2007 Nov;50(5):926-32
2-(butyryl-(2'-(4-fluoro-5-methylisoxazol-3-ylsulfamoyl)biphenyl-4-ylmethyl)amino)-N-isopropyl-3-methylbutyramide  0   *Isoxazoles *Sulfonamides Receptors, Angiotensin/antagonists & inhibitors Receptor, Endothelin A/antagonists & inhibitors. Drug Metab Dispos 2007 May;35(5):795-805
2-(butyryl-(2'-(4-chloro-5-methylisoxazol-3-ylsulfamoyl)biphenyl-4-ylmethyl)amino)-N-isopropyl-3-methylbutyramide  0   *Isoxazoles *Sulfonamides Receptors, Angiotensin/antagonists & inhibitors Receptor, Endothelin A/antagonists & inhibitors. Drug Metab Dispos 2007 May;35(5):795-805
2-(butyryl-(2'-(4,5-dimethylisoxazol-3-ylsulfamoyl)biphenyl-4-ylmethyl)amino)-N-isopropyl-3-methylbutyramide  0   *Isoxazoles *Sulfonamides Receptors, Angiotensin/antagonists & inhibitors Receptor, Endothelin A/antagonists & inhibitors. Drug Metab Dispos 2007 May;35(5):795-805
N-butyloxycarbonyl-2-(4-imidazol-1-ylmethylphenyl)-4-butoxybenzenesulfonamide  0   *Sulfonamides Receptors, Angiotensin/agonists. J Med Chem 2006 Nov 30;49(24):7160-8
N-butyloxycarbonyl-3-(4-imidazol-1-ylmethylphenyl)-5-propylthiophene-2-sulfonamide  0   *Sulfonamides *Thiophenes Receptors, Angiotensin/agonists. J Med Chem 2006 Nov 30;49(24):7160-8
Dear1 protein, mouse  0   *Receptors, Angiotensin *Receptors, Endothelin. Physiol Genomics 2005 Nov 17;23(3):257-68
2-methylsulfanyl-3-(2'-(2H-tetrazol-5-yl)biphenyl-4-ylmethyl)-3H-quinazolin-4-one  0   *Quinazolines *Tetrazoles Receptors, Angiotensin/antagonists & inhibitors. J Med Chem 2006 Mar 9;49(5):1526-35
Nalp6 protein, rat  0   *Receptors, Angiotensin *Receptors, Vasopressin. Nat Med 1995 Oct;1(10):1074-81
AGTRAP protein, human  0   *Adaptor Proteins, Signal Transducing Receptors, Angiotensin. Int J Biochem Cell Biol 2002 Jan;34(1):93-102
pyrazolidine-3,5-dione  0   *Pyrazoles Receptors, Angiotensin. Acta Crystallogr C 2001 Nov;57(Pt 11):1330-2
dimethyl (1-methyl-1,3-benzimidazol-5-yl)aminomethylenepropanedioate  0   *Benzimidazoles *Cinnamates Receptors, Angiotensin/antagonists & inhibitors. Acta Crystallogr C 2000 Aug;56( Pt 8):1007-8
sarcosine(1)-angiotensin II receptor  0   *Receptors, Angiotensin. Neuroscience 2000;95(4):981-91
SL 910102-90 DL  0   *Pyrimidines *Tetrazoles Receptors, Angiotensin/antagonists & inhibitors. J Pharm Biomed Anal 1998 May;17(1):111-24
L 163017  0   *Imidazoles *Pyridines Receptors, Angiotensin/antagonists & inhibitors. Eur J Pharmacol 1995 Dec 29;294(2-3):439-50
L 163082  0   *Imidazoles *Sulfonamides Receptors, Angiotensin/antagonists & inhibitors. Circulation 1996 Mar 1;93(5):1009-19
L 159913  0   *Triazoles Receptors, Angiotensin/antagonists & inhibitors. Clin Exp Hypertens 1995 Aug;17(6):931-53
L 163958  0   *Biphenyl Compounds *Triazoles Receptors, Angiotensin/antagonists & inhibitors. J Med Chem 1995 Sep 15;38(19):3741-58
XR 510  0   *Biphenyl Compounds *Imidazoles Receptors, Angiotensin/antagonists & inhibitors. J Med Chem 1995 Jul 21;38(15):2938-45
AT4 receptor  0   *Receptors, Angiotensin. Peptides 1994;15(6):1037-44

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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012

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