encyclopedia of medical concepts
ψ 
ψ 

Octreotide

More information in Books or onNLM PubMed
Definition: A potent, long-acting synthetic SOMATOSTATIN octapeptide analog that inhibits secretion of GROWTH HORMONE and is used to treat hormone-secreting tumors; DIABETES MELLITUS; HYPOTENSION, ORTHOSTATIC; HYPERINSULINISM; hypergastrinemia; and small bowel fistula.     
Pharmacological Action Antineoplastic Agents, Hormonal; Gastrointestinal Agents
Other names Octreotide Acetate; Sandoz 201995; Sandoz 201 995; SMS 201995; SMS 201 995; SM 201995; SM 201 995; SAN 201995; SAN 201 995; Compound 201995; Compound 201 995; Sandoz 201-995; Sandostatine; Sandostatin; SMS 201-995; SM 201-995; SAN 201-995; Octreotide Acetate Salt; Compound 201-995Drugs* : SANDOSTATIN; SANDOSTATIN LAR; OCTREOTIDE ACETATE; OCTREOTIDE ACETATE (PRESERVATIVE FREE)
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
177Lu-octreotate  0   Octreotide/*analogs & derivatives Lutetium. Eur J Nucl Med Mol Imaging 2007 Aug;34(8):1219-27
68Ga-octreotide, DOTA(0)-Tyr(3)  0   *Organometallic Compounds Octreotide/*analogs & derivatives Gallium Radioisotopes. Endocr Relat Cancer 2010 Mar;17(1):R53-73
sandostatinLAR  0   Octreotide/*analogs & derivatives. Neuroendocrinology 2009;89(3):296-301
90Y-octreotate, DOTA(0)-Tyr(3)-Thr(8)  0   *Organometallic Compounds Octreotide/*analogs & derivatives Yttrium Radioisotopes. Nucl Med Rev Cent East Eur 2008;11(1):5-11
technetium Tc 99m hydrazinonicotinyl-Tyr(3)-Thr(8)-octreotide  0   *Organotechnetium Compounds Octreotide/*analogs & derivatives. J Nucl Med 2008 Jul;49(7):1060-5
technetium Tc 99m (EDDA-HYNIC)octreotate  0   *Organotechnetium Compounds Octreotide/*analogs & derivatives. Eur J Nucl Med Mol Imaging 2007 Oct;34(10):1545-55
(technetium 99m-EDDA-tricine-HYNIC(0)-Nal(1)-Thr(8))octreotide  0   *Organotechnetium Compounds Octreotide/*analogs & derivatives. Nucl Med Biol 2007 Aug;34(6):651-7
yttrium cyclohexyldiethylenetriaminepentaacetic acid-octreotide  0   Pentetic Acid/*analogs & derivatives Octreotide/*analogs & derivatives Yttrium Radioisotopes. J Med Chem 2006 Jul 13;49(14):4297-304
111In-DOTA-TOC  0   Octreotide/*analogs & derivatives Indium Radioisotopes. Eur J Nucl Med Mol Imaging 2005 Oct;32(10):1144-51
177Lu-octreotide, DOTA(0)-Tyr(3)  0   Octreotide/*analogs & derivatives Lutetium. J Nucl Med 2005 Aug;46(8):1310-6
111In-octreotate, DOTA(0)-Tyr(3)-Thr(8)  0   *Organometallic Compounds Octreotide/*analogs & derivatives Indium Radioisotopes. Eur J Nucl Med Mol Imaging 2004 Sep;31(9):1257-62
Ga(III)-DOTATOC  0   *Organometallic Compounds Octreotide/*analogs & derivatives Gallium Radioisotopes. J Med Chem 2005 Mar 10;48(5):1506-14
111In-octreotide, DTPA(0)  0   Pentetic Acid/*analogs & derivatives Octreotide/*analogs & derivatives Indium Radioisotopes. J Nucl Med 2005 Jan;46 Suppl 1:62S-6S
90Y-octreotide, DOTA-Tyr(3)  0   Octreotide/*analogs & derivatives Yttrium Radioisotopes. Nucl Med Biol 2004 Aug;31(6):821-4
99mTc-octreotide  0   *Organotechnetium Compounds Octreotide/*analogs & derivatives. Nucl Med Biol. 2004 Feb;31(2):231-9
DOTA-Tyr(1)-octreotate  0   *Heterocyclic Compounds, 1-Ring Octreotide/*analogs & derivatives. Bioconjug Chem 2002 Jul-Aug;13(4):721-8
Y-DOTAGA-tate  0   Octreotide/*analogs & derivatives. Cancer Biother Radiopharm 2002 Oct;17(5):527-33
Y-DOTA-t-GA-tate  0   Octreotide/*analogs & derivatives. Cancer Biother Radiopharm 2002 Oct;17(5):527-33
(177lutetium-DOTA(O)Tyr3)octreotate  0   *Organometallic Compounds Octreotide/*analogs & derivatives Lutetium. Eur J Nucl Med 2001 Sep;28(9):1319-25
octreotate, maltotriose-iodotyrosyl(3)  0   *Trisaccharides Octreotide/*analogs & derivatives Iodine Radioisotopes. Eur J Nucl Med 2002 Jan;29(1):28-38
copper 1,4,8,11--tetraazacyclotetradecane-N,N',N'',N'''-tetraacetic acid-octreotide  0   *Organometallic Compounds Octreotide/*analogs & derivatives Copper Radioisotopes. J Nucl Med 2001 Feb;42(2):213-21
technetium Tc 99m-tricine-hydrazinonicotinyl-Phe(1)-Tyr(3)-octreotide  0   *Organotechnetium Compounds Octreotide/*analogs & derivatives. Eur J Nucl Med 2000 Jun;27(6):628-37
octreotide-conjugated paclitaxel  0   *Octreotide *Taxoids. Chem Biol. 2000 Jul;7(7):453-61
technetium Tc 99m hydrazinonicotinyl-Tyr(3)-octreotide  0   *Organotechnetium Compounds Octreotide/*analogs & derivatives. J Nucl Med 2000 Jun;41(6):1114-9
copper-1,4,8,11-tetraazacyclotetradecane-N,N',N'',N'''-tetraacetic acid-octreotate  0   *Organometallic Compounds Octreotide/*analogs & derivatives. Clin Cancer Res 1999 Nov;5(11):3608-16
octreotide, DOTA-Tyr(3)  0   Octreotide/*analogs & derivatives. Eur J Nucl Med 1999 Jul;26(7):693-8
technetium Tc 99m cyclopentadienyltricarbonyloctreotide  0   *Organotechnetium Compounds Octreotide. Nucl Med Biol 1999 Jan;26(1):1-7
octreotide, DOTA-Phe(1)  0   *Heterocyclic Compounds, 1-Ring Octreotide/*analogs & derivatives. Bioorg Med Chem Lett 1998 May 19;8(10):1207-10
octreotide, iodoTyr(3)  0   Octreotide/*analogs & derivatives Iodine Radioisotopes. Eur J Pharmacol 1998 May 8;348(2-3):311-20
SDZ 223228  178181-50-5   Octreotide/*analogs & derivatives Fluorine Radioisotopes. Nucl Med Biol 1997 Aug;21(6):819-25
(DOTA(0)-Phe(1)-Tyr(3))octreotide  0   Octreotide/*analogs & derivatives Indium Radioisotopes Yttrium Radioisotopes.
Pharma Action Radiopharmaceuticals
Eur J Nucl Med;1997 Apr;24(4):368-71
DTPA-benzyl-acetamido-D-Phe(1),Tyr(3)-octreotide  0   Pentetic Acid/*analogs & derivatives Octreotide/*analogs & derivatives. Digestion 1996;57 Suppl 1:17-21
octreotide, CPTA-Phe(1)  0   Octreotide/*analogs & derivatives. J Nucl Med 1995 Dec;36(12):2315-25
octreotide, TETA-Phe(1)  0   Octreotide/*analogs & derivatives. J Nucl Med 1995 Dec;36(12):2315-25
indium-111-octreotide  0   Octreotide/*analogs & derivatives Indium Radioisotopes.
Pharma Action Radiopharmaceuticals
J Nucl Biol Med 1994 Dec;38(4):576-8
(PnAO-(D)Phe(1))octreotide  0   Octreotide/*analogs & derivatives. Eur J Nucl Med 1994 May;21(5):437-44
SDZ CO 611  119719-11-8 L-Cysteinamide, N-(1-deoxy-4-O-alpha-D-glucopyranosyl-D-fructopyranos-1-yl)-D-phenylalanyl-L-cysteinyl-L-phenylalanyl-D-tryptophyl-L-lysyl-L-threonyl-N-(2-hydroxy-1-(hydroxymethyl)propyl)-, cyclic (2-7)-disulfide, (R-(R*,R*))  Octreotide/*analogs & derivatives. Life Sci 1993;53(6):517-25
desferrioxamine B-succinyl-phenylalanine(1)-octreotide  151956-24-0   Deferoxamine/*analogs & derivatives Octreotide/*analogs & derivatives Gallium Radioisotopes. Horm Metab Res Suppl 1993;27:12-7
technetium Tc 99m 6-(4-thioureabenzyl)-3,3,9,9-tetramethyl-4,8-diazaundecane-phenylalanine(1)-octreotide  151956-25-1   *Organotechnetium Compounds Octreotide/*analogs & derivatives. Horm Metab Res Suppl 1993;27:12-7
4-nitrobenzo-2-oxa-1,3-diazol-octreotide  0   4-Chloro-7-nitrobenzofurazan/*analogs & derivatives Octreotide/*analogs & derivatives. Br J Pharmacol 1993 Feb;108(2):298-303
EE 581  141949-00-0   *Azides Octreotide/*analogs & derivatives. Endocrinology 1992 May;130(5):2937-46
phenylalanyl-cysteinyl-tyrosyl-tryptophyl-lysyl-threonyl-cysteinyl-N-naphthylalanine amide  138248-87-0   Octreotide/*analogs & derivatives. Am J Physiol 1992 Mar;262(3 Pt 1):G432-8
SDZ 215-811  142694-57-3   Pentetic Acid/*analogs & derivatives Octreotide/*analogs & derivatives Indium Radioisotopes Terbium.
Pharma Action Radiopharmaceuticals
Life Sci 1991;49(22):1583
SDZ 204-090  96608-80-9   Octreotide/*analogs & derivatives. Biochem J 1990;265(1):39
RC 121  99660-13-6   Octreotide/*analogs & derivatives. Life Sci 1987;41(8):1011
3-Tyr-octreotide  103667-46-5   Octreotide/*analogs & derivatives. Life Sci 1985;36(19):1829

To share this definition, click "text" (Facebook, Twitter) or "link" (blog, mail) then paste text link
Ads by Google

Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012

Warning: the drugs or drug combinations referred to here may be similar or related, but are not be the same ones and may not have the same pharmacological action as other substances described on the same page or in the same row. Please refer to product monograph or to your doctor
This website is accredited by Health On the Net Foundation. Click to verify.
We comply with the HONcode standard for trustworthy health information: verify here.
About Reference.MD Privacy