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Receptors, Bradykinin

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Definition: Cell surface receptors that bind BRADYKININ and related KININS with high affinity and trigger intracellular changes which influence the behavior of cells. The identified receptor types (B-1 and B-2, or BK-1 and BK-2) recognize endogenous KALLIDIN; t-kinins; and certain bradykinin fragments as well as bradykinin itself.  note specific subtypes; DF: RECEPT BRADYKININ   
Examples Receptor, Bradykinin B1; Receptor, Bradykinin B2 		Other names Bradykinin Receptors; Receptor, Bradykinin; Bradykinin Receptor
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
3-benzyl-1-(4-guanidinylphenyl)-4-phenyl-2H-1,4-benzodiazepin-2-one  0   *Benzodiazepinones *Guanidines Receptors, Bradykinin/antagonists & inhibitors. Peptides 2001 Sep;22(9):1397-402
martinellic acid  0   *Pyrroles *Quinolines Receptors, Bradykinin/antagonists & inhibitors. Org Lett 2001 Jul 12;3(14):2189-91
Pam-Lys(0)-Arg(1)-Pro(2)-Pro(3)-Gly(4)-Phe(5)-Ser(6)-Pro(7)-Phe(8)-Arg(9)-OH  0   *Lipopeptides Receptors, Bradykinin/agonists. Biopolymers 2001 Apr 15;58(5):511-20
Pam-Gly(-1)-Lys(0)-Arg(1)-Pro(2)-Pro(3)-Gly(4)-Phe(5)-Ser(6)-Pro(7)-Phe(8)-Arg(9)-OH  0   *Lipopeptides Bradykinin/*analogs & derivatives Receptors, Bradykinin/agonists. Biopolymers 2001 Apr 15;58(5):511-20
JMV 1640  0   *Oligopeptides *Thiazepines Receptors, Bradykinin/antagonists & inhibitors. J Med Chem 2000 Jun 15;43(12):2387-94
bradyzide  0   *Pyrrolidines *Thiosemicarbazones Receptors, Bradykinin/antagonists & inhibitors. Br J Pharmacol 2000 Jan;129(1):77-86
N-(4-(2-(2-((2-dmethylaminoethyl)methylamino)ethylaminocarbonyl)pyrrolidinylsulfonyl)-2-nitrophenylamino)-N'-diphenylmethylthiourea  0   Proline/*analogs & derivatives Thiourea/*analogs & derivatives Receptors, Bradykinin/antagonists & inhibitors. J Med Chem 2000 Mar 9;43(5):769-71
J 324  0   *Peptides, Cyclic Receptors, Bradykinin/antagonists & inhibitors. J Pept Res 2000 Jan;55(1):63-71
B6014  0   *Oligopeptides Receptors, Bradykinin/agonists. Hypertension 2000 Jan;35(1 Pt 1):32-7
LF 16-0687  0   *Quinolines Receptors, Bradykinin/antagonists & inhibitors. Immunopharmacology 1999 Sep;43(2-3):187-94
JMV 1465  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/agonists. J Med Chem 1999 Oct 7;42(20):4193-201
JMV 1609  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/agonists. J Med Chem 1999 Oct 7;42(20):4193-201
arginyl-prolyl-prolyl--glycyl-phenylalanyl-seryl-(3S)(amino)-5-(carbonylmethyl)-2,3-dihydro-1,5-benzothiazepin-4(5H)-one-arginine  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/agonists. J Med Chem 1999 Oct 7;42(20):4185-92
JMV 1116  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/agonists. J Med Chem 1999 Oct 7;42(20):4185-92
B 9430  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/antagonists & inhibitors. Eur J Pharmacol 1999 Jul 2;376(1-2):83-9
B 9858  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/antagonists & inhibitors. Eur J Pharmacol 1999 Jul 2;376(1-2):83-9
R 715  0   Bradykinin/*analogs & derivatives Receptors, Bradykinin/antagonists & inhibitors. Neuroscience 1999;92(3):1043-9
MEN 11270  0   *Oligopeptides *Peptides, Cyclic Receptors, Bradykinin/antagonists & inhibitors. J Pharmacol Exp Ther 1999 Jun;289(3):1250-6
LF 16.0335  0   *Amidines *Piperazines Receptors, Bradykinin/antagonists & inhibitors. Br J Pharmacol 1998 Sep;125(2):365-72
FR 193517  0   *Aminopyridines *Quinolines Receptors, Bradykinin/antagonists & inhibitors. J Med Chem 1998 Nov 5;41(23):4587-98
FR 184280  0   *Pyridines *Quinolines Receptors, Bradykinin/antagonists & inhibitors. J Med Chem 1998 Oct 8;41(21):4062-79
FR 165649  0   *Quinolines Receptors, Bradykinin/antagonists & inhibitors. Br J Pharmacol 1998 Jun;124(3):441-6
CP 0597  0   *Oligopeptides Receptors, Bradykinin/antagonists & inhibitors. Stroke 1997 Jul;28(7):1430-6
FR 190997  0   *Quinolines Receptors, Bradykinin/agonists. Mol Pharmacol 1997 Jul;52(1):16-20
FR 167344  0   *Pyridines Receptors, Bradykinin/antagonists & inhibitors. Mol Pharmacol 1997 Feb;51(2):171-6
FR 173657  0   *Quinolines Receptors, Bradykinin/antagonists & inhibitors.
Pharma Action Anti-Inflammatory Agents, Non-Steroidal 		Hypertension 1997 Apr;29(4):951-6
NPC 18688  0   *Imidazoles *Spiro Compounds Receptors, Bradykinin/antagonists & inhibitors. J Med Chem 1996 Aug 2;39(16):3169-73
NPC 18521  0   *Imidazoles *Spiro Compounds Receptors, Bradykinin/antagonists & inhibitors. J Med Chem 1996 Aug 2;39(16):3169-73
bradykinin, Lys-Leu(8)-desArg(9)  0   Kallidin/*analogs & derivatives Receptors, Bradykinin/antagonists & inhibitors. J Pharmacol Exp Ther 1993 Jul;266(1):192-9
kallidin receptor  0   *Receptors, Bradykinin. Agents Actions Suppl 1992;38 ( Pt 2):382-89
deltibant  140661-97-8   *Peptides Receptors, Bradykinin/antagonists & inhibitors. Lancet 1991;338(8773):1011
icatibant  130308-48-4   Bradykinin/*analogs & derivatives Receptors, Bradykinin/antagonists & inhibitors.
Pharma Action Adrenergic beta-Antagonists ; Anti-Inflammatory Agents, Non-Steroidal 		Eur J Pharmacol 1990;182(2):395FIRAZYR

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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012
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