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Excitatory Amino Acid Antagonists
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Definition
: Drugs that bind to but do not activate excitatory amino acid receptors, thereby blocking the actions of agonists.
GEN or unspecified; prefer specifics; DF: EAA ANTAG
Other names
Receptor Antagonists, Glutamate; Antagonists, Glutamate Receptor; Antagonists, Glutamate; Antagonists, EAA; Glutamate Receptor Antagonists; EAA Antagonists; Antagonists, Excitatory Amino Acid; Amino Acid Antagonists, Excitatory; Glutamate Antagonists; Amino Acids, Excitatory, Antagonists
Substances having this pharmacologic action:
ifenprodil
;
2,3-piperidinedicarboxylic acid
;
2-amino-7-phosphonoheptanoic acid
;
gabapentin
;
HA 966
;
caroverine
;
2-amino-3-phosphonopropionic acid
;
Dizocilpine Maleate
;
Kynurenic Acid
;
6-Cyano-7-nitroquinoxaline-2,3-dione
;
2-Aminoadipic Acid
;
2-Amino-5-phosphonovalerate
;
Riluzole
;
Memantine
;
Phencyclidine
;
Phenobarbital
;
Ibogaine
;
Ketamine
;
Dextromethorphan
;
Dextrorphan
;
glutamic acid diethyl ester
;
ketobemidone
;
LY 341495
;
6-methyl-2-(phenylethynyl)pyridine
;
licostinel
;
L 701324
;
1-aminoindan-1,5-dicarboxylic acid
;
GV 150526A
;
3,5-dihydroxyphenylglycine
;
GYKI 53655
;
4-carboxyphenylglycine
;
alpha-methyl-4-carboxyphenylglycine
;
aptiganel
;
6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-quinoxalinedione
;
LY 235959
;
CGP 39653
;
gacyclidine
;
4-trans-2-carboxy-5,7-dichloro-4-phenylaminocarbonylamino-1,2,3,4-tetrahydroquinoline
;
NPC 12626
;
GYKI 52466
;
HU 211
;
2,3-dioxo-6-nitro-7-sulfamoylbenzo(f)quinoxaline
;
conantokin-T
;
2-amino-4-methyl-5-phosphono-3-pentenoic acid
;
CGP 39551
;
SDZ EAA 494
;
5,7-dichlorokynurenic acid
;
selfotel
;
conotoxin GV
;
FG 9041
;
7-chlorokynurenic acid
;
eliprodil
;
carbinoxamine, dextromethorphan, pseudoephedrine drug combination
;
3-(2-carboxypiperazin-4-yl)propyl-1-phosphonic acid
Substance
CAS Registry & name
Categories
Source
Drugs
*
lamotrigine
84057-84-1
*Triazines
Analgesics
Bipolar Disorder
Cleft Lip
Excitatory Amino Acid Antagonists
Antimanic Agents.
Pharma Action
Anticonvulsants
;
Calcium Channel Blockers
Br J Clin Pharmacol 1985;20(6):619
LAMICTAL CD
;
LAMICTAL
;
LAMOTRIGINE
;
LAMICTAL XR
;
LAMICTAL ODT