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Receptor, Bradykinin B2

More information in Books or onNLM PubMed
Definition: A constitutively expressed subtype of bradykinin receptor that may play a role in the acute phase of the inflammatory and pain response. It has high specificity for intact forms of BRADYKININ and KALLIDIN. The receptor is coupled to G-PROTEIN, GQ-G11 ALPHA FAMILY and G-PROTEIN, GI-GO ALPHA FAMILY signaling proteins.      Other names Receptors, Bradykinin B2; B2 Receptors, Bradykinin; B2 Receptor, Bradykinin; Receptor, Bradykinin Type 2; Bradykinin B2 Receptors; Bradykinin Type 2 Receptor; Bradykinin B2 Receptor
 
SubstanceCAS Registry & nameCategoriesSourceDrugs*
helokinestatin  0   *Venoms Receptor, Bradykinin B2/antagonists & inhibitors. Peptides 2008 Jan;29(1):65-72
N-(2-(4-(2-amino-5-(dimethylamino)pentanoyl)piperazin-1-yl)-1,1-dimethyl-2-oxoethyl)-2,3-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonamide  0   *Quinolines *Sulfonamides Receptor, Bradykinin B2/antagonists & inhibitors. J Med Chem 2006 Jun 15;49(12):3602-13
2-(3-oxo-1-(toluene-4-sulfonyl)-1,2,3,4-4H-quinoxalin-2-yl)-N-phenyl-acetamide  0   *Acetanilides *Tosyl Compounds Receptor, Bradykinin B2/antagonists & inhibitors Receptor, Bradykinin B1/antagonists & inhibitors. Biol Chem 2006 Feb;387(2):189-94
(4-amino-5-(4-(4-(2,4-dichloro-3-(2,4-dimethyl-8-quinolyloxymethyl)phenylsulfonamido)tetrahydro-2H-4-pyranoylcarbonyl)piperazino)-5-oxopentyl)(trimethyl)ammonium  0   *Sulfonamides Ornithine/*analogs & derivatives Receptor, Bradykinin B2/antagonists & inhibitors. J Pharmacol Exp Ther 2005 Nov;315(2):616-23
bradykinin, Hyp(3)-TyrMe(8)  0   Bradykinin/*analogs & derivatives Receptor, Bradykinin B2/agonists. Methods Find Exp Clin Pharmacol 2004 May;26(4):247-52

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Sources: NLM Medical Subject Headings, NIH UMLS, Drugs@FDA, FDA AERS original data copyright United States Government. No endorsement implied. Last modified 6/6/2012
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