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CGP 39653

under 2-Amino-5-phosphonovalerate
More information in Books or onNLM PubMed
More on 2-Amino-5-phosphonovalerate Definition: The D-enantiomer is a potent and specific antagonist of NMDA glutamate receptors (RECEPTORS, N-METHYL-D-ASPARTATE). The L form is inactive at NMDA receptors but may affect the AP4 (2-amino-4-phosphonobutyrate; APB) excitatory amino acid receptors.      Other names 2 Amino 5 phosphonopentanoate; dl-APV; d-APV; 5-Phosphononorvaline; 2-Amino-5-phosphonopentanoate; 2-Amino-5-phosphonovaleric Acid; 2-Amino-5-phosphonopentanoic Acid; 2-APV; 5 Phosphononorvaline; 2 Amino 5 phosphonovaleric Acid; 2 Amino 5 phosphonovalerate; 2 Amino 5 phosphonopentanoic Acid
SubstanceCAS Registry & nameCategoriesSourceDrugs*
CGP 39653 [ 2-amino-4-propyl-5-phosphono-3-pentenoic acid,CGP-39653 ]
  NMDA receptor antagonist; structure given in first source 		132472-31-2 3-Heptenoic acid, 2-amino-4-(phosphonomethyl)-, (E)-(+-)  2-Amino-5-phosphonovalerate/*analogs & derivatives
Pharma Action Excitatory Amino Acid Antagonists 		Eur J Pharmacol 1991;192(1):19

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