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Enkephalin, Ala(2)-MePhe(4)-Gly(5)-
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Definition
: An enkephalin analog that selectively binds to the MU OPIOID RECEPTOR. It is used as a model for drug permeability experiments.
Pharmacological Action
Analgesics, Opioid
;
Anti-Arrhythmia Agents
;
Neurotransmitter Agents
Other names
DAGO; DAGOL; RX 783006; Enkephalin, D-
Ala2-
NMe-
Phe4-
Gly-
ol; D Ala2 NMe Phe4 Gly ol Enkephalin; 2 Ala 4 MePhe 5 Gly Enkephalin; Tyr-
Ala-
Gly-
(NMe)Phe-
Gly-
ol; RX-
783006; Enkephalin, alanyl(2)-
methylphenylalanyl(4)-
glycin; DAMGE; D-
Ala2-
NMe-
Phe4-
Gly-
ol Enkephalin; Ala(2)-
MePhe(4)-
Gly-
ol(5) Enkephalin; 2-
Ala-
4-
MePhe-
5-
Gly-
Enkephalin; DAMGO; D-
Ala(2)-
MePhe(4)-
Gly-
ol(5) Enkephalin
Substance
CAS Registry & name
Categories
Source
Drugs
*
enkephalin, Ala(2)-
MePhe(4)-
GlyNH2(5)
0
Enkephalin, Ala(2)-MePhe(4)-Gly(5)-/*analogs & derivatives.
Peptides 2006 Jun;27(6):1507-13