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HIV Fusion Inhibitors
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Definition
: Inhibitors of the fusion of HIV to host cells, preventing viral entry. This includes compounds that block attachment of HIV ENVELOPE PROTEIN GP120 to CD4 RECEPTORS.
See Also
Membrane Fusion
Other names
Entry Inhibitors, HIV; HIV Cell Fusion Inhibitors; HIV Entry Inhibitors; Fusion Inhibitors, HIV
Substances having this pharmacologic action:
enfuvirtide
Substance
CAS Registry & name
Categories
Source
Drugs
*
Qadirvirtide
0
*Peptides
HIV Fusion Inhibitors.
Pak J Pharm Sci. 2011 Oct;24(4):593-5
BMS-
488043
0
*Piperazines
HIV Fusion Inhibitors.
J Virol 2006 Apr;80(8):4017-25
TAK-
220
0
*Piperidines
HIV Fusion Inhibitors.
Antimicrob Agents Chemother. 2005 Nov;49(11):4708-15
maraviroc
0
*Cyclohexanes
*Triazoles
Receptors, CCR5/antagonists & inhibitors
HIV Fusion Inhibitors.
Drug Metab Dispos. 2005 Apr;33(4):587-95
SELZENTRY
873140 compound
0
*Benzoates
*Piperazines
*Spiro Compounds
HIV Fusion Inhibitors.
Mol Pharmacol 2005 Apr;67(4):1268-82
TNX-
355
0
*Antibodies, Monoclonal
HIV Fusion Inhibitors.
AIDS Patient Care STDS. 2003 Dec;17(12):655
BMS-
378806
0
*Piperazines
HIV Fusion Inhibitors.
J Virol 2003 Oct;77(19):10528-36
PRO-
140 monclonal antibody
0
*HIV Antibodies
*Antibodies, Monoclonal, Humanized
Anti-HIV Agents
Receptors, CCR5
HIV Fusion Inhibitors.
Aids Patient Care STDS 2000 Dec;14(12):671; IDrugs. 2001 Sep;4(9):1068-71
TAK 779
229005-80-5
*Amides
*Quaternary Ammonium Compounds
Receptors, CCR5/antagonists & inhibitors
HIV Fusion Inhibitors.
Proc Natl Acad Sci U S A 1999 May 11;96(10):5698-703
CD4-
IgG(2)
0
*CD4 Immunoadhesins
HIV-1
HIV Fusion Inhibitors.
AIDS Res Hum Retroviruses 1995 May;11(5):533-9
JM 3100
155148-31-5
*Heterocyclic Compounds
Receptors, CXCR4/antagonists & inhibitors
HIV Fusion Inhibitors.
Pharma Action
Anti-HIV Agents
Antimicrob Agents Chemother 1994 Apr;38(4):668-74
MOZOBIL