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| HIV Fusion Inhibitors |
| Inhibitors of the fusion of HIV to host cells, preventing viral entry. This includes compounds that block attachment of HIV ENVELOPE PROTEIN GP120 to CD4 RECEPTORS.
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See Also Membrane Fusion | Other names HIV Entry Inhibitors; Fusion Inhibitors, HIV; Entry Inhibitors, HIV; HIV Cell Fusion Inhibitors; HIV Entry Inhibitors; Fusion Inhibitors, HIV
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| Substances having this pharmacologic action: enfuvirtide
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| Substance | CAS Registry & name | Categories | Source | Drugs*
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| JM 3100
| 155148-31-5
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*Heterocyclic Compounds HIV Fusion Inhibitors Receptors, CXCR4/antagonists & inhibitors.
Pharma Action Anti-HIV Agents
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Antimicrob Agents Chemother 1994 Apr;38(4):668-74
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| TAK 779
| 229005-80-5
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*Amides *Quaternary Ammonium Compounds Receptors, CCR5/antagonists & inhibitors HIV Fusion Inhibitors.
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Proc Natl Acad Sci U S A 1999 May 11;96(10):5698-703
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CD4-IgG(2)
| 0
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*CD4 Immunoadhesins HIV-1 HIV Fusion Inhibitors.
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AIDS Res Hum Retroviruses 1995 May;11(5):533-9
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BMS-378806
| 0
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HIV Fusion Inhibitors *Piperazines.
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J Virol 2003 Oct;77(19):10528-36
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4,4-difluoro-N-((1S)-3-(exo-3-(3-isopropyl-5-methyl-4H-1,2,4-triazol-4-yl)-8-azabicyclo(3.2.1)oct-8-yl)-1-phenylpropyl)cyclohexanecarboxamide
| 0
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Receptors, CCR5/antagonists & inhibitors HIV Fusion Inhibitors *Cyclohexanes *Triazoles.
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Drug Metab Dispos. 2005 Apr;33(4):587-95
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| PRO 140
| 0
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Anti-HIV Agents Receptors, CCR5 HIV Fusion Inhibitors *Antibodies, Monoclonal *HIV Antibodies.
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Aids Patient Care STDS 2000 Dec;14(12):671; IDrugs. 2001 Sep;4(9):1068-71
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| 873140 compound
| 0
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HIV Fusion Inhibitors *Benzoates *Piperazines *Spiro Compounds.
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Mol Pharmacol 2005 Apr;67(4):1268-82
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TNX-355
| 0
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HIV Fusion Inhibitors *Antibodies, Monoclonal.
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AIDS Patient Care STDS. 2003 Dec;17(12):655
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TAK-220
| 0
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HIV Fusion Inhibitors *Piperidines.
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Antimicrob Agents Chemother. 2005 Nov;49(11):4708-15
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BMS-488043
| 0
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HIV Fusion Inhibitors *Piperazines.
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J Virol 2006 Apr;80(8):4017-25
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