encyclopedia of medical concepts
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Excitatory Amino Acid Transporter 1
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Definition
: A glial type glutamate plasma membrane transporter protein found predominately in ASTROCYTES. It is also expressed in HEART and SKELETAL MUSCLE and in the PLACENTA.
Other names
Transporter, SLC1A3; GLAST 1 Glutamate Aspartate Transporter; EAAT 1 Excitatory Amino Acid Transporter; Glutamate Aspartate Transporter 1; GLAST-
1 Glutamate Aspartate Transporter; EAAT-
1 Excitatory Amino Acid Transporter; SLC1A3 Transporter
Substance
CAS Registry & name
Categories
Source
Drugs
*
2-
amino-
4-
(4-
methoxyphenyl)-
7-
(naphthalen-
1-
yl)-
5-
oxo-
5,6,7,8-
tetrahydro-
4H-
chromene-
3-
carbonitrile
0
*Benzopyrans
Excitatory Amino Acid Transporter 1/antagonists & inhibitors.
J Med Chem 2010 Oct 14;53(19):7180-91
3-
azabicyclo(3.3.0)octane-
4,6-
dicarboxylic acid
0
*Dicarboxylic Acids
*Bicyclo Compounds, Heterocyclic
Excitatory Amino Acid Transporter 1/antagonists & inhibitors
Excitatory Amino Acid Transporter 2/antagonists & inhibitors
Excitatory Amino Acid Transporter 3/antagonists & inhibitors.
J Med Chem 2006 Jan 12;49(1):172-8
SLC1A3 protein, human
0
*Excitatory Amino Acid Transporter 1.
Slc1a3 protein, mouse
0
*Excitatory Amino Acid Transporter 1.
Slc1a3 protein, rat
0
*Excitatory Amino Acid Transporter 1.