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Receptors, Lysophosphatidic Acid
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Definition
: A subfamily of lysophospholipid receptors with specificity for LYSOPHOSPHATIDIC ACIDS.
Other names
LPA 1 Receptor; Edg 7 Receptor; Edg 4 Receptor; Acid Receptors, Lysophosphatidic; Acid Receptor, Lysophosphatidic; vzg-
1 Receptor; edg-
2 Receptor; Receptor, Lysophosphatidic Acid; LPA3 Receptor; LPA2 Receptor; LPA1 Receptor; LPA-
1 Receptor; LPA Receptors; Edg4 Protein; Edg2 Protein; Edg-
7 Receptor; Edg-
4 Receptor; EDG7 Protein; vzg 1 Receptor; edg 2 Receptor
Substance
CAS Registry & name
Categories
Source
Drugs
*
Lpa5 protein, rat
0
*Receptors, Lysophosphatidic Acid.
Mol Carcinog 2011 Aug;50(8):635-42
phosphoric acid mono-
(3-
(4-
benzyloxyphenyl)-
2-
octadec-
9-
enoylaminopropyl) ester
0
*Oleic Acids
*Phosphoric Acid Esters
Receptors, Lysophosphatidic Acid/antagonists & inhibitors.
Oncol Rep 2010 Dec;24(6):1515-20
(4'-
(4-
(1-
(2-
chlorophenyl)ethoxycarbonylamino)-
3-
methylisoxazol-
5-
yl)biphenyl-
4-
yl)acetic acid
0
*Carbamates
*Phenylacetates
Receptors, Lysophosphatidic Acid/antagonists & inhibitors.
Br J Pharmacol 2010 Aug;160(7):1699-713
LPAR5 protein, mouse
0
*Receptors, Lysophosphatidic Acid.
Gastroenterology. 2010 Feb;138(2):649-58
LPAR6 protein, human
0
*Receptors, Lysophosphatidic Acid.
Prostaglandins Other Lipid Mediat 2009 Sep;89(3-4):57-65
GPR87 protein, mouse
0
*Receptors, Lysophosphatidic Acid.
Biochem Biophys Res Commun 2007 Nov 23;363(3):861-6
GPR87 protein, human
0
*Receptors, Lysophosphatidic Acid.
Biochem Biophys Res Commun 2007 Nov 23;363(3):861-6
LPAR5 protein, human
0
*Receptors, Lysophosphatidic Acid.
J Pharmacol Exp Ther 2006 Aug;318(2):619-28
tetradecyl phosphonate
0
*Fatty Alcohols
*Phosphonic Acids
Receptors, Lysophosphatidic Acid/antagonists & inhibitors.
J Med Chem 2005 Jul 28;48(15):4919-30
oleoyl thiophosphate
0
*Fatty Alcohols
*Phosphoric Acid Esters
Receptors, Lysophosphatidic Acid/agonists.
J Med Chem 2005 Jul 28;48(15):4919-30
GPR45 protein, human
0
*Receptors, Lysophosphatidic Acid.