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G-Protein-Coupled Receptor Kinases
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Definition
: A family of serine-threonine kinases that are specific for G-PROTEIN-COUPLED RECEPTORS. They are regulatory proteins that play a role in G-protein-coupled receptor densensitization.
Examples
beta-Adrenergic Receptor Kinases
;
G-Protein-Coupled Receptor Kinase 1
;
G-Protein-Coupled Receptor Kinase 4
;
G-Protein-Coupled Receptor Kinase 5
Other names
Receptor Kinases, G-
Protein-
Coupled; Kinases, G-
Protein-
Coupled Receptor; G Protein Coupled Receptor Kinases
Substance
CAS Registry & name
Categories
Source
Drugs
*
GRK7 protein, zebrafish
EC 2.7.1.17
*G-Protein-Coupled Receptor Kinases.
Neuron 2005 Jul 21;47(2):231-42
GRK7 protein, human
EC 2.7.1.15
*G-Protein-Coupled Receptor Kinases.
FEBS Lett 1998 Mar 13;424(3):159-64
G-
protein-
coupled receptor kinase 6
EC 2.7.11.16
*G-Protein-Coupled Receptor Kinases
Receptors, G-Protein-Coupled.
J Biol Chem 1994 Sep 9;269(36):22691-7