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Cysteine Proteinase Inhibitors
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Definition
: Exogenous and endogenous compounds which inhibit CYSTEINE ENDOPEPTIDASES.
/biosyn /physiol permitted only with endogenous proteinase inhib; DF: CYSTEINE PROTEINASE INHIB
Other names
Cysteine Proteinase Inhibitors, Exogenous; Cysteine Proteinase Inhibitors, Endogenous; Cysteine Proteinase Antagonists; Cysteine Protease Inhibitors; alpha Cysteine Protease Inhibitors; Proteinase Inhibitors, Cysteine; Proteinase Antagonists, Cysteine; Protease Inhibitors, alpha-
Cysteine; Protease Inhibitors, Cysteine; Inhibitors, alpha-
Cysteine Protease; Inhibitors, Cysteine Proteinase; Inhibitors, Cysteine Protease; Antagonists, Cysteine Proteinase; alpha-
Cysteine Protease Inhibitors; Acid Cysteine Proteinase Inhibitors
Substances having this pharmacologic action:
benzyloxycarbonylphenylalanylalanine diazomethyl ketone
;
E 64
;
4-hydroxy-2-nonenal
;
leupeptin
;
calpastatin
;
calpain inhibitors
;
phenylalanyl-prolyl-arginine-chloromethyl ketone
;
geldanamycin
;
Cystatin B
;
Salivary Cystatins
;
benzyloxycarbonyl-isoleucyl-glutamyl(O-tert-butyl)-alanyl-leucinal
;
Kininogens
;
Cystatins
;
BIRC5 protein, human
;
aloxistatin
;
aspartyl-glutamyl-valyl-aspartal
;
benzoylcarbonyl-aspartyl-glutamyl-valyl-aspartyl-fluoromethyl ketone
;
Ac-aspartyl-glutamyl-valyl-aspartyl-aminomethylcoumarin
;
benzyloxycarbonyl-isoleucyl-glutamyl-threonyl-aspartic acid fluoromethyl ketone
;
L 709049
;
benzyloxycarbonylvalyl-alanyl-aspartyl fluoromethyl ketone
;
N-acetyl-tyrosyl-valyl-alanyl-aspartyl chloromethyl ketone
;
clasto-lactacystin beta-lactone
;
acetyl-aspartyl-glutamyl-valyl-aspartal
;
cystatin, egg-white
;
nitroaspirin
;
butyloxycarbonyl-O-methyl-aspartyl-fluoromethyl ketone
;
inhibitor of apoptosis, Nucleopolyhedrovirus
;
lactacystin
;
N-(3-propylcarbamoyloxirane-2-carbonyl)-isoleucyl-proline
;
N-acetylleucyl-leucyl-methioninal
;
calpeptin
;
benzyloxycarbonylleucyl-leucyl-leucine aldehyde
;
acetylleucyl-leucyl-norleucinal
;
MDL 201053
;
calpain inhibitor III
Substance
CAS Registry & name
Categories
Source
Drugs
*
interleukin-
1beta-
converting enzyme inhibitor
96282-35-8
*Viral Proteins
*Serpins
Cysteine Proteinase Inhibitors.
Cell 1992 May 15;69(4):597-604
ovocystatin
0
Peptides
Cysteine Proteinase Inhibitors.
Microbiol Immunol 1991;35(7):583-8