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ψ
ψ
Receptors, GABA-B
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Definition
: A subset of GABA RECEPTORS that signal through their interaction with HETEROTRIMERIC G-PROTEINS.
Other names
GABA-
B Receptors; Baclofen Receptors; Receptors, GABA B; Receptor, GABA-
B; Receptor, Baclofen; GABA B Receptors; GABA B Receptor; Receptors, Baclofen; GABA-
B Receptor; Baclofen Receptor
Substance
CAS Registry & name
Categories
Source
Drugs
*
N-
(bicyclo(2.2.1)hept-
2-
yl)-
2-
methyl-
5-
(4-
(trifluoromethyl)phenyl)-
4-
pyrimidinamine
0
*Norbornanes
*Pyrimidines
Receptors, GABA-B
GABA Modulators.
Psychopharmacology (Berl) 2011 May;215(1):117-28
3-
amino-
2-
hydroxypropylcyclohexylmethylphosphinic acid
0
*Phosphinic Acids
Receptors, GABA-B/antagonists & inhibitors.
Br J Pharmacol 2006 Nov;149(5):581-90
Gabbr2 protein, mouse
0
*Receptors, GABA-B.
GABBR2 protein, human
0
*Receptors, GABA-B.
CGP 13501
0
*Phenols
Receptors, GABA-B/agonists.
Mol Pharmacol 2001 Nov;60(5):963-71
CGP 7930
0
*Phenols
Receptors, GABA-B/agonists.
Mol Pharmacol 2001 Nov;60(5):963-71
5-
amino-
3-
(4-
chlophenyl)pentanoic acid
0
Baclofen/*analogs & derivatives
Receptors, GABA-B.
Eur J Pharmacol 2001 Apr 13;417(3):177-80
CGP 47332A
0
*Phosphinic Acids
Receptors, GABA-B/antagonists & inhibitors.
Eur J Pharmacol 1999 Oct 27;383(2):137-41
3-
aminopropyl-
(1,1,-
difluoro-
n-
butyl)phosphinic acid
0
*Phosphinic Acids
Receptors, GABA-B/antagonists & inhibitors.
Eur J Pharmacol 1999 Jun 25;374(3):351-4
3-
aminopropyl-
P-
(alpha-
hydroxybenzyl)phosphinic acid
0
*Phosphinic Acids
Receptors, GABA-B/antagonists & inhibitors.
Eur J Pharmacol 1999 Jun 25;374(3):351-4
Gabbr2 protein, rat
0
*Receptors, GABA-B.
Genomics 1999 Mar 15;56(3):288-95; Nature 1998 Dec 17;396(6712):674-9; Science 1999 Jan 1;283(5398):74-7
4-
hydroxy-
4-
(4'-
chlorophenyl)hexanamide
0
*Amides
Receptors, GABA-B/antagonists & inhibitors.
Arzneimittelforschung 1998 Aug;48(8):797-801
3-
hydroxy-
3-
(4'-
chlorophenyl)pentanamide
0
*Amides
Receptors, GABA-B/antagonists & inhibitors.
Arzneimittelforschung 1998 Aug;48(8):797-801
2-
hydroxy-
2-
(4'-
chlorophenyl)butyramide
0
*Amides
Receptors, GABA-B/antagonists & inhibitors.
Arzneimittelforschung 1998 Aug;48(8):797-801
CGP 44532
0
*Phosphinic Acids
gamma-Aminobutyric Acid/*analogs & derivatives
Receptors, GABA-B/agonists.
Life Sci 1998;62(17-18):1525-30
CGP 61334
0
*Phosphinic Acids
*Benzoic Acids
Receptors, GABA-B/antagonists & inhibitors.
Eur J Pharmacol 1997 Feb 5;320(1):9-13
(3-
(1-
((3-
(cyclohexylmethyl)hydroxyphosphinyl)-
2-
hydroxypropyl)amino)ethyl)benzoic acid
153994-81-1
*Phosphinic Acids
*Benzoic Acids
Receptors, GABA-B/antagonists & inhibitors.
Eur J Pharmacol 1997 Feb 5;320(1):9-13
GABA type B receptor, subunit 1
0
*Receptors, GABA-B.
Nature 1997 Mar 20;386(6622):239-46
CGP 71872
0
*Azides
*Organophosphorus Compounds
Iodine Radioisotopes
Receptors, GABA-B/antagonists & inhibitors.
Nature 1997 Mar 20;386(6622):239-46