encyclopedia of medical concepts
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raf Kinases
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Definition
: A family of closely-related serine-threonine kinases that were originally identified as the cellular homologs of the retrovirus-derived V-RAF KINASES. They are MAP kinase kinase kinases that play important roles in SIGNAL TRANSDUCTION.
Examples
Oncogene Proteins v-raf
;
Proto-Oncogene Proteins B-raf
;
Proto-Oncogene Proteins c-raf
Other names
raf Serine Theonine Protein Kinases; raf Proto Oncogene Proteins; mil raf Protein Kinases; Proto-
Oncogene Proteins, raf; Proto Oncogene Proteins raf; Proteins raf, Proto-
Oncogene; Protein Kinases, mil-
raf; MIL RAF Proteins; Kinases, raf; Kinases, mil-
raf Protein; raf Serine-
Theonine Protein Kinases; raf Proto-
Oncogene Proteins; Proto-
Oncogene Proteins raf; raf MAP Kinase Kinase Kinases; mil-
raf Protein Kinases; MIL-
RAF Proteins
Substance
CAS Registry & name
Categories
Source
Drugs
*
LBT 613
0
*Isoquinolines
raf Kinases/antagonists & inhibitors.
Clin Cancer Res 2006 Mar 15;12(6):1785-93
AAL 881
0
*Isoquinolines
raf Kinases/antagonists & inhibitors.
Clin Cancer Res 2006 Mar 15;12(6):1785-93
sorafenib
0
*Benzenesulfonates
*Pyridines
Receptors, Vascular Endothelial Growth Factor
raf Kinases.
Pharma Action
Antineoplastic Agents
;
Protein Kinase Inhibitors
Curr Pharm Des 2002;8(25):2249-53
NEXAVAR
lin-
45 protein, C elegans
EC 2.7.1.-
*Caenorhabditis elegans Proteins
*raf Kinases
Signal Transduction
Proto-Oncogene Proteins c-raf.
Nature 1993 May 13;363(6425):133-40