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Receptors, Lysosphingolipid
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Definition
: A subfamily of lysophospholipid receptors with specificity for LYSOSPHINGOLIPIDS such as sphingosine-1-phosphate and sphingosine phosphorylcholine.
Other names
edg 8 Protein; edg 6 Receptor; edg 3 Protein; edg 1 Receptor; Sphingosine 1 Phosphate Receptors; Sphingosine 1 Phosphate Receptor; Receptors, Sphingosine-
1-
Phosphate; edg 1 Protein; Receptors, Sphingosine Phosphorylcholine; Receptors, Edg; Receptor, edg-
6; Receptor, edg-
1; Receptor, Sphingosine 1 Phosphate; Receptor, S1P5; Receptor, S1P4; Receptor, S1P3; Receptor, S1P2; Receptor, Nrg-
1; Receptor, Edg-
5; Protein, edg-
8
Substance
CAS Registry & name
Categories
Source
Drugs
*
sphingosine-
1-
phosphate receptor-
2, rat
0
*Receptors, Lysosphingolipid.
Hepatology. 2012 Jan;55(1):267-76
CS 0777
0
*Amino Alcohols
*Pyrroles
Receptors, Lysosphingolipid.
J Clin Pharmacol. 2009 Jan;49(1):50-62.
spingosine-
1-
phosphate receptor 4, mouse
0
*Receptors, Lysosphingolipid.
J Immunol. 2002 Oct 15;169(8):4084-7.
5-
(3-
(2-
(2-
hydroxy-
1-
(hydroxymethyl)ethyl)-
5-
methyl-
1,2,3,4-
tetrahydro-
6-
isoquinolinyl)-
1,2,4-
oxadiazol-
5-
yl)-
2-
((1-
methylethyl)oxy)benzonitrile
0
*Isoquinolines
*Oxadiazoles
Receptors, Lysosphingolipid/agonists.
J Med Chem. 2011 Oct 13;54(19):6724-33.
1-
(hydroxymethyl)-
3-
(3-
octylphenyl)cyclobutane
0
*Benzene Derivatives
*Cyclobutanes
Receptors, Lysosphingolipid/antagonists & inhibitors.
J Pharmacol Exp Ther 2011 Sep;338(3):879-89
S1pr1 protein, mouse
0
*Receptors, Lysosphingolipid.
J Bone Miner Metab. 2010 Nov;28(6):659-71
5-
(3-
chloro-
4-
(2,3-
dihydroxy-
propoxy)benzylidene)-
2-
propylimino-
3-
o-
tolyl-
thiazolidin-
4-
one
0
*Thiazoles
Receptors, Lysosphingolipid/antagonists & inhibitors.
J Med Chem 2010 May 27;53(10):4198-211
2-
amino-
2-
(2-
(2'-
fluoro-
4'-
(4-
methylphenylthio)biphenyl-
4-
yl)ethyl)propane-
1,3-
diol
0
*Biphenyl Compounds
*Propanolamines
Receptors, Lysosphingolipid/agonists.
J Med Chem 2010 Apr 22;53(8):3154-68
sphingosine-
1-
phosphate receptor-
2, mouse
0
*Receptors, Lysosphingolipid.
Stroke 2008 Dec;39(12):3411-7
AUY 954
0
*Thiophenes
beta-Alanine/*analogs & derivatives
Receptors, Lysosphingolipid/agonists.
Chem Biol 2006 Nov;13(11):1227-34
1-
(4-
((4-
phenyl-
5-
trifluoromethyl-
2-
thienyl)methoxy)benzyl)azetidine-
3-
carboxylic acid
0
*Azetidines
*Thiophenes
Receptors, Lysosphingolipid/agonists.
Drug Metab Dispos 2006 Aug;34(8):1367-75
3-
amino-
4-
(3-
hexylphenylamino)-
4-
oxobutylphosphonic acid
0
*Anilides
*Phosphonic Acids
Receptors, Lysosphingolipid/antagonists & inhibitors.
Nat Chem Biol 2006 Aug;2(8):434-41
Edg3 protein, mouse
0
*Receptors, Lysosphingolipid.
Circulation 2004 Nov 23;110(21):3355-9
S1PR2 protein, human
0
*Receptors, Lysosphingolipid.
J Biol Chem 2003 Aug 29;278(35):32841-51
S1PR1 protein, human
0
*Receptors, Lysosphingolipid.
Cancer Res. 2003 Aug 15;63(16):5151-8