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Metalloendopeptidases
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Definition
: ENDOPEPTIDASES which use a metal such as ZINC in the catalytic mechanism.
Examples
Botulinum Toxins
;
Collagenases
;
Gelatinases
;
Insulysin
;
Lysostaphin
;
Matrix Metalloproteinases
;
Neprilysin
;
PHEX Phosphate Regulating Neutral Endopeptidase
;
Pregnancy-Associated Plasma Protein-A
;
Procollagen N-Endopeptidase
;
Pronase
;
Thermolysin
Other names
Metalloendopeptidase; Metallo-
Endoproteinases
Substance
CAS Registry & name
Categories
Source
Drugs
*
SAK-
RGD-
K2-
Hirul
EC 3.4.24.-
*Hirudins
*Metalloendopeptidases
*Recombinant Fusion Proteins.
Acta Biochim Pol. 2009;56(1):41-53.
NRD1 protein, human
EC 3.4.24.61
*Metalloendopeptidases
Alcohol-Related Disorders.
J Psychiatr Res. 2011 Nov;45(11):1419-25
stromal processing peptidase, Arabidopsis
EC 3.4.24.-
*Metalloendopeptidases
*Arabidopsis Proteins
Chloroplast Proteins.
PLoS One. 2011;6(8):e23039.
BlaR1 protein, Staphylococcus aureus
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases
Membrane Proteins
Intracellular Signaling Peptides and Proteins.
Antimicrob Agents Chemother. 1993 May;37(5):1144-9.
Pitrm1 protein, mouse
EC 3.4.24.-
*Metalloendopeptidases.
Dev Dyn 20009 Dec;238(12):3175-84
Afg3l1 protein, mouse
EC 3.4.24.-
*Metalloendopeptidases.
Genomics 2001 Aug;76(1-3):58-65
staphylokinase SFH
EC 3.4.24.-
*Metalloendopeptidases
*Recombinant Fusion Proteins.
J Thromb Thrombolysis 2007 Dec;24(3):283-92
S2P metalloprotease, Methanocaldococcus jannaschii
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases.
Science. 2007 Dec 7;318(5856):1608-12
SAK-
RGD-
K2-
Hir
0
*Hirudins
*Metalloendopeptidases
*Recombinant Fusion Proteins.
Thromb Haemost 2007 Jun;97(6):1037-45
VAP2 protein, Crotalus atrox
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
Eur J Biochem 1998 Apr 1;253(1):36-41
DPY-
31 protein, C elegans
EC 3.4.-
*Metalloendopeptidases
*Caenorhabditis elegans Proteins.
Genetics 2004 Nov;168(3):259-73
halysase, Gloydius halys
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
J Biochem (Tokyo) 2003 Nov;134(5):739-49
berythractivase, Bothrops erythromelas
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
Biol Chem 2005 Apr;386(4):369-74
Ste23 protein, S cerevisiae
EC 3.4.24.-
*Metalloendopeptidases
*Saccharomyces cerevisiae Proteins.
J Biol Chem 2005 Jul 29;280(30):27481-90
ADAMTS13 protein, mouse
EC 3.4.24.-
*Metalloendopeptidases.
J Thromb Haemost 2005 May;3(5):1064-73
ZmpA protein, Burkholderia cenocepacia
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases.
J Bacteriol 2005 Jul;187(13):4421-9
invadolysin, human
EC 3.4.24.-
*Metalloendopeptidases.
J Cell Biol 2004 Nov 22;167(4):673-86
invadolysin, Drosophila
EC 3.4.24.-
*Metalloendopeptidases
*Drosophila Proteins.
J Cell Biol 2004 Nov 22;167(4):673-86
BjussuMP-
I
EC 3.4.24.-
*Metalloendopeptidases
Snake Venoms.
Toxicon. 2004 Aug;44(2):215-23
ECEL1 protein, human
EC 3.4.24.-
*Metalloendopeptidases.
Ecel1 protein, rat
EC 3.4.24.-
*Metalloendopeptidases.
MMP23A protein, human
EC 3.4.24.-
*Metalloendopeptidases.
Spg7 protein, mouse
EC 3.4.24.-
*Metalloendopeptidases.
dactylysin, Xenopus
EC 3.5.24.60
*Metalloendopeptidases
*Xenopus Proteins.
Comp Biochem Physiol B Biochem Mol Biol. 2002 Aug;132(4):751-9
STE24 protein, S cerevisiae
EC 3.4.24.-
*Membrane Proteins
*Metalloendopeptidases
*Saccharomyces cerevisiae Proteins.
Zmpste24 protein, mouse
EC 3.4.24.-
*Membrane Proteins
*Metalloendopeptidases.
chloroplast processing enzyme protein, Arabidopsis
EC 3.4.24.-
*Metalloendopeptidases
*Arabidopsis Proteins
Protein Processing, Post-Translational.
Kae1 protein, S cerevisiae
EC 3.4.24.-
*Metalloendopeptidases
*Saccharomyces cerevisiae Proteins.
Biochem J 2004 Jan 15;377(Pt 2):395-405
ProB protein, Ehrlichia canis
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases.
DNA Seq 2003 Apr;14(2):109-21
ProA protein, Ehrlichia canis
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases.
DNA Seq 2003 Apr;14(2):109-21
AmpA protein, Dictyostelium protozoan
EC 3.4.24.-
*Metalloendopeptidases
*Protozoan Proteins.
J Muscle Res Cell Motil. 2002;23(7-8):817-28
ZmpC protein, Streptococcus pneumoniae
EC 3.4.24.-
*Metalloendopeptidases.
Mol Microbiol 2003 Aug;49(3):795-805
halydin protein, Gloydius halys
EC 3.4.24.-
*Metalloendopeptidases.
Biochem Biophys Res Commun 2003 Sep 26;309(3):637-42
basparin A, Bothrops asper
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
Arch Biochem Biophys 2003 Oct 1;418(1):13-24
molecule metalloprotease-
related protein-
1, human
EC 3.4.24.-
*Metalloendopeptidases.
DNA Res 2003 Jun 30;10(3);123-8
factor X activator, Russell's viper
EC 3.4.24.-
*Metalloendopeptidases
*Viper Venoms.
Haemostasis 2001 May-Dec;31(3-6):
factor X activator, Vipera lebetina
EC 3.4.24.-
*Metalloendopeptidases
*Viper Venoms.
Haemostasis 2001 May-Dec;31(3-6):123-32
UNC-
71 protein, C elegans
EC 3.4.24.-
*Metalloendopeptidases
*Caenorhabditis elegans Proteins
Disintegrins.
Development 2003 Jul;130(14):3147-61
xolloid-
related protein, Xenopus
EC 3.4.24.-
*Metalloendopeptidases.
Mech Dev 2002 Dec;119(2);177-90
FACE-
2 protein, C elegans
EC 3.4.22.-
*Metalloendopeptidases
*Caenorhabditis elegans Proteins.
Biochem J 2003 Mar 15;370(Pt 3):1047-54
FACE-
1 protein, C elegans
EC 3.4.22.-
*Caenorhabditis elegans Proteins
*Metalloendopeptidases.
Biochem J 2003 Mar 15;370(Pt 3):1047-54
agkistin, Agkistrodon halys
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
Biochem Biophys Res Commun 2003 Feb 7;301(2):298-303
bothropasin, Bothrops jararaca
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
Toxicon 2003 Feb;41(2):217-27
Mop protein, Vibrio cholerae
EC 3.4.24.-
*Metalloendopeptidases.
Infect Immun 2003 Jan;71(1):510-5
TM-
3 protein, Trimeresurus mucrosquamatus
EC 3.4.24.-
*Crotalid Venoms
*Metalloendopeptidases.
Acta Crystallogr D Biol Crystallogr 2002 Jul;58(Pt 7):1118-28
mikarin
EC 3.4.24.-
*Elapid Venoms
*Metalloendopeptidases.
Arch Biochem Biophys 2002 Dec 1;408(1):87-92
hemorrhagic toxin HR-
1a, Trimeresurus flavoviridis
EC 3.4.24.-
*Metalloendopeptidases
*Viper Venoms.
Toxicon 2002 Sep;40(9):1369-75
Rri1 protein, S cerevisiae
EC 3.4.24.-
*Metalloendopeptidases
*Saccharomyces cerevisiae Proteins.
Science 2002 Oct 18;298(5593):608-11
VfpA protein, Vibrio fluvialis
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases.
Microb Pathog 2002 Sep;33(3):127-34
StcE protein, E coli
EC 3.4.24.-
*Metalloendopeptidases
*Escherichia coli Proteins.
Mol Microbiol 2002 Jul;45(2):277-88
testase 4, human
EC 3.4.24.-
*Metalloendopeptidases.
Gene 2002 Apr 17;288(1-2):203-10
PEGylated staphylokinase SY161
EC 3.4.24.-
*Metalloendopeptidases
*Polyethylene Glycols.
J Pharm Biomed Anal 2002 Jun 1;28(5):953-63
InhA2 protein, Bacillus thuringiensis
EC 3.4.24.-
*Bacterial Proteins
*Metalloendopeptidases.
J Bacteriol 2002 Jun;184(12):3296-304
MTP-
1 protein, Ancylostoma caninum
EC 3.4.24.-
*Metalloendopeptidases.
Mol Biochem Parasitol 2002 Apr 9;120(2):291-6
N(4)-
(2,2-
dimethyl-
1-
methylcarbamoylpropyl)-
N(1)-
hydroxy-
2-
hydroxymethyl-
3-
(4-
methoxyphenyl)succinamide
0
*Hydroxamic Acids
Metalloendopeptidases/antagonists & inhibitors
Matrix Metalloproteinases/antagonists & inhibitors.
J Med Chem 2002 May 23;45(11):2289-93
Adt-
1 protein, C elegans
0
*Metalloendopeptidases
*Caenorhabditis elegans Proteins.
J Biol Chem 2002 Apr 5;277(14):12228-36
AG3433
0
*Furans
*Nitriles
*Pyrroles
Metalloendopeptidases/antagonists & inhibitors.
J Org Chem 2002 Mar 8;67(5):1699-702
MEP-
1 protein, Ancylostoma caninum
EC 3.4.24.-
*Metalloendopeptidases
*Helminth Proteins.
Mol Biochem Parasitol 2002 Jan;119(1):107-16
BB 3644
0
*Aminopyridines
*Hydroxamic Acids
Metalloendopeptidases/antagonists & inhibitors.
Int J Cancer 2002 Mar 10;98(2):210-5
N-
hydroxy-
2-
((2,2-
difluoroethoxy)(4-
methoxyphenyl)phosphoryl)-
1,2,3,4-
tetrahydroisoquinoline-
3-
carboxamide
0
*Hydroxylamines
*Tetrahydroisoquinolines
Metalloendopeptidases/antagonists & inhibitors.
J Med Chem 2002 Feb 14;45(4):930-6
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