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Receptors, Angiotensin
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Definition
: Cell surface proteins that bind ANGIOTENSINS and trigger intracellular changes influencing the behavior of cells.
note specific subtypes; do not confuse receptors that bind to ANGIOTENSIN II and ANGIOTENSIN III with specific angiotensin receptor subtypes
Examples
Receptor, Angiotensin, Type 1
;
Receptor, Angiotensin, Type 2
Other names
Angiotensin Receptors; Receptor, Angiotensin III; Receptor, Angiotensin II; Angiotensin III Receptor; Angiotensin II Receptor
Substance
CAS Registry & name
Categories
Source
Drugs
*
N-
butyloxycarbonyl-
3-
(4-
(2-
oxopyrrolidin-
1-
ylmethyl)phenyl)-
5-
isobutylthiophene-
2-
sulfonamide
0
*Sulfonamides
*Thiophenes
Receptors, Angiotensin/agonists.
Bioorg Med Chem 2010 Jun 15;18(12):4570-90
3-
(1-
biphenyl-
4-
ylmethyl-
3-
ethoxycarbonyl-
1-
butylcarbamoyl)propionate-
3'-
methyl-
2'-
(pentanoyl(2'-
(tetrazol-
5-
ylate)biphenyl-
4'-
ylmethyl)amino)butyrate
0
*Aminobutyric Acids
*Tetrazoles
Receptors, Angiotensin/antagonists & inhibitors
Neprilysin/antagonists & inhibitors.
Lancet 2010 Apr 10;375(9722):1255-66
Agtrap protein, rat
0
*Receptors, Angiotensin.
Hypertension 2007 Nov;50(5):926-32
2-
(butyryl-
(2'-
(4-
fluoro-
5-
methylisoxazol-
3-
ylsulfamoyl)biphenyl-
4-
ylmethyl)amino)-
N-
isopropyl-
3-
methylbutyramide
0
*Isoxazoles
*Sulfonamides
Receptors, Angiotensin/antagonists & inhibitors
Receptor, Endothelin A/antagonists & inhibitors.
Drug Metab Dispos 2007 May;35(5):795-805
2-
(butyryl-
(2'-
(4-
chloro-
5-
methylisoxazol-
3-
ylsulfamoyl)biphenyl-
4-
ylmethyl)amino)-
N-
isopropyl-
3-
methylbutyramide
0
*Isoxazoles
*Sulfonamides
Receptors, Angiotensin/antagonists & inhibitors
Receptor, Endothelin A/antagonists & inhibitors.
Drug Metab Dispos 2007 May;35(5):795-805
2-
(butyryl-
(2'-
(4,5-
dimethylisoxazol-
3-
ylsulfamoyl)biphenyl-
4-
ylmethyl)amino)-
N-
isopropyl-
3-
methylbutyramide
0
*Isoxazoles
*Sulfonamides
Receptors, Angiotensin/antagonists & inhibitors
Receptor, Endothelin A/antagonists & inhibitors.
Drug Metab Dispos 2007 May;35(5):795-805
N-
butyloxycarbonyl-
2-
(4-
imidazol-
1-
ylmethylphenyl)-
4-
butoxybenzenesulfonamide
0
*Sulfonamides
Receptors, Angiotensin/agonists.
J Med Chem 2006 Nov 30;49(24):7160-8
N-
butyloxycarbonyl-
3-
(4-
imidazol-
1-
ylmethylphenyl)-
5-
propylthiophene-
2-
sulfonamide
0
*Sulfonamides
*Thiophenes
Receptors, Angiotensin/agonists.
J Med Chem 2006 Nov 30;49(24):7160-8
Dear1 protein, mouse
0
*Receptors, Angiotensin
*Receptors, Endothelin.
Physiol Genomics 2005 Nov 17;23(3):257-68
2-
methylsulfanyl-
3-
(2'-
(2H-
tetrazol-
5-
yl)biphenyl-
4-
ylmethyl)-
3H-
quinazolin-
4-
one
0
*Quinazolines
*Tetrazoles
Receptors, Angiotensin/antagonists & inhibitors.
J Med Chem 2006 Mar 9;49(5):1526-35
Nalp6 protein, rat
0
*Receptors, Angiotensin
*Receptors, Vasopressin.
Nat Med 1995 Oct;1(10):1074-81
AGTRAP protein, human
0
*Adaptor Proteins, Signal Transducing
Receptors, Angiotensin.
Int J Biochem Cell Biol 2002 Jan;34(1):93-102
pyrazolidine-
3,5-
dione
0
*Pyrazoles
Receptors, Angiotensin.
Acta Crystallogr C 2001 Nov;57(Pt 11):1330-2
dimethyl (1-
methyl-
1,3-
benzimidazol-
5-
yl)aminomethylenepropanedioate
0
*Benzimidazoles
*Cinnamates
Receptors, Angiotensin/antagonists & inhibitors.
Acta Crystallogr C 2000 Aug;56( Pt 8):1007-8
sarcosine(1)-
angiotensin II receptor
0
*Receptors, Angiotensin.
Neuroscience 2000;95(4):981-91
SL 910102-
90 DL
0
*Pyrimidines
*Tetrazoles
Receptors, Angiotensin/antagonists & inhibitors.
J Pharm Biomed Anal 1998 May;17(1):111-24
L 163017
0
*Imidazoles
*Pyridines
Receptors, Angiotensin/antagonists & inhibitors.
Eur J Pharmacol 1995 Dec 29;294(2-3):439-50
L 163082
0
*Imidazoles
*Sulfonamides
Receptors, Angiotensin/antagonists & inhibitors.
Circulation 1996 Mar 1;93(5):1009-19
L 159913
0
*Triazoles
Receptors, Angiotensin/antagonists & inhibitors.
Clin Exp Hypertens 1995 Aug;17(6):931-53
L 163958
0
*Biphenyl Compounds
*Triazoles
Receptors, Angiotensin/antagonists & inhibitors.
J Med Chem 1995 Sep 15;38(19):3741-58
XR 510
0
*Biphenyl Compounds
*Imidazoles
Receptors, Angiotensin/antagonists & inhibitors.
J Med Chem 1995 Jul 21;38(15):2938-45
AT4 receptor
0
*Receptors, Angiotensin.
Peptides 1994;15(6):1037-44