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Drug Resistance, Multiple
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Definition
: Simultaneous resistance to several structurally and functionally distinct drugs.
DRUG RESISTANCE, MULTIPLE, BACTERIAL; DRUG RESISTANCE, MULTIPLE, VIRAL; and DRUG RESISTANCE, MULTIPLE, FUNGAL are also available
See Also
Genes, MDR
;
Multidrug Resistance-Associated Proteins
;
P-Glycoproteins
Examples
Drug Resistance, Multiple, Bacterial
;
Drug Resistance, Multiple, Fungal
;
Drug Resistance, Multiple, Viral
Other names
Multidrug Resistance; Resistance, Multiple Drug; Multiple Drug Resistance; Multi-
Drug Resistance
Substance
CAS Registry & name
Categories
Source
murucoidin V
0
*Glycosides
Drug Resistance, Multiple/drug effects.
J Nat Prod. 2012 Jan 27;75(1):93-7
small multidrug-
resistance pump, Staphylococcus aureus
0
*Antiporters
Drug Resistance, Multiple.
J Biol Chem 1994 Nov 25;269(47):29998-30004
2-
(N-
(4-
methoxyphenylethylaminocarbonyl))-
5-
hydroxychromone
0
*Chromones
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 2005 Nov 17;48(23):7275-81
2-
(N-
(3,4-
dimethoxyphenylethylaminocarbonyl))-
5-
hydroxychromone
0
*Chromones
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 2005 Nov 17;48(23):7275-81
2-
(4-
n-
butylpiperazin-
1-
ylcarbonyl)-
5-
hydroxychromone
0
*Chromones
*Piperazines
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 2005 Nov 17;48(23):7275-81
Abcc5 protein, mouse
0
*Multidrug Resistance-Associated Proteins
Drug Resistance, Multiple.
ATMRP5 protein, Arabidopsis
0
*Multidrug Resistance-Associated Proteins
*Arabidopsis Proteins
Drug Resistance, Multiple.
Abcc4 protein, rat
0
*Multidrug Resistance-Associated Proteins
Drug Resistance, Multiple.
ArpC protein, Pseudomonas putida
0
*Bacterial Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
Microbiology 2001 Jan;147(Pt 1):43-51
ArpB protein, Pseudomonas putida
0
*Bacterial Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
Microbiology 2001 Jan;147(Pt 1):43-51
ArpA protein, Pseudomonas putida
0
*Bacterial Proteins
*Carrier Proteins
Drug Resistance, Multiple.
Microbiology 2001 Jan;147(Pt 1):43-51
TtgI protein, Pseudomonas putida
0
*Bacterial Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
J Bacteriol 2001 Jul;183(13):3967-73
POHL protein, marine sponge
0
*Trans-Activators
Drug Resistance, Multiple.
Environ Toxicol Chem 2001 Jan;20(1):198-204
multidrug resistance-
associated protein 1
0
*Multidrug Resistance-Associated Proteins
Drug Resistance, Multiple.
4-
deacetoxyagosterol
0
*Sterols
Drug Resistance, Multiple.
Bioorg Med Chem Lett 2000 Nov 20;10(22):2521-4
7-
O-
benzoylpyripyropene A
0
*Pyridones
*Sesquiterpenes
Drug Resistance, Multiple.
J Antibiot (Tokyo) 2000 Oct;53(10):1201-6
FLU1 protein, Candida albicans
0
*Fungal Proteins
*Drug Resistance, Multiple
*ATP-Binding Cassette Transporters.
Microbiology 2000 Nov;146 ( Pt 11):2743-54
RAB6C protein, human
EC 3.6.1.-
*rab GTP-Binding Proteins
Drug Resistance, Multiple.
Gene 2000 Oct 17;257(1):67-75
R 101933
0
*Benzazepines
*Quinolines
Drug Resistance, Multiple
P-Glycoprotein/antagonists & inhibitors.
Clin Cancer Res 2000 Apr;6(4):1365-71
OC 144-
093
0
*Imidazoles
Drug Resistance, Multiple.
Cancer Res 2000 Jun 1;60(11):2964-72
doxorubicin-
gallium-
transferrin conjugate
0
*Doxorubicin
*Organometallic Compounds
*Transferrin
Gallium
Drug Resistance, Multiple.
Anticancer Res 2000 Mar-Apr;20(2A):799-808
MEF1 protein, human
0
*DNA-Binding Proteins
*Transcription Factors
Genes, MDR
Drug Resistance, Multiple.
Biochemistry 2000 Jan 11;39(1):194-204
CP 147673
0
*Piperazines
Drug Resistance, Multiple
P-Glycoprotein/antagonists & inhibitors.
Biochemistry 2000 Jan 11;39(1):75-85
CP 172732
0
*Piperazines
*Thiazoles
Drug Resistance, Multiple
P-Glycoprotein/antagonists & inhibitors.
Biochemistry 2000 Jan 11;39(1):75-85
CP 162398
0
*Piperazines
*Quinolines
Drug Resistance, Multiple
P-Glycoprotein/antagonists & inhibitors.
Biochemistry 2000 Jan 11;39(1):75-85
MexXY protein, Pseudomonas aeruginosa
0
*Bacterial Proteins
Drug Resistance, Multiple.
Antimicrob Agents Chemother 1999 Nov;43(11):2624-8
LY 329146
0
*Sulfonamides
*Thiophenes
Drug Resistance, Multiple.
Bioorg Med Chem Lett 1999 Dec 6;9(23):3381-6
B 4121
0
Clofazimine/*analogs & derivatives
Drug Resistance, Multiple.
Oncol Rep 2000 Jan-Feb;7(1):193-5
tariquidar
206873-63-4
*Quinolines
Drug Resistance, Multiple.
Br J Pharmacol 1999 Sep;128(2):403-11
ABCC5 protein, human
0
*Multidrug Resistance-Associated Proteins
Drug Resistance, Multiple.
Cancer Res 1997 Aug 15;57(16):3537-47
9-
hydroxy-
2-
(2-
(dimethylamino)ethyl)-
6-
((2-
(dimethylamino)ethyl)amino)-
2,3-
dihydro-
1H,7H-
pyrimido(5,6,1-
de)acridine-
1,3,7-
trione
0
*Acridines
*Pyrimidinones
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 1999 Jul 15;42(14):2535-41
9-
amino-
2-
(2-
(dimethylamino)ethyl)-
6-
((2-
(dimethylamino)ethyl)amino)-
2,3-
dihydro-
1H,7H-
pyrimido(5,6,1-
de)acridine-
1,3,7-
trione
0
*Acridines
*Pyrimidinones
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 1999 Jul 15;42(14):2535-41
6-
((2-
aminoethyl)amino)-
2-
(2-
(dimethylamino)ethyl)-
2,3-
dihydro-
1H,7H-
pyrimido(5,6,1-
de)acridine-
1,3,7-
trione
0
*Acridines
*Pyrimidinones
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 1999 Jul 15;42(14):2535-41
reversin 205
0
*Oligopeptides
Drug Resistance, Multiple.
Biochem Pharmacol 1999 Aug 15;58(4):571-86
reversin 121
0
*Oligopeptides
Drug Resistance, Multiple.
Biochem Pharmacol 1999 Aug 15;58(4):571-86
MM 36
0
*Anisoles
*Nitriles
Drug Resistance, Multiple
Drug Resistance, Neoplasm.
J Med Chem 1999 May 20;42(10):1687-97
multidrug resistance-
associated protein 2
0
*Multidrug Resistance-Associated Proteins
Jaundice, Chronic Idiopathic
Drug Resistance, Multiple.
Mol Pharmacol 1999 May;55(5):929-37
MexA protein, Pseudomonas aeruginosa
0
*Bacterial Outer Membrane Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
J Bacteriol 1993 Nov;175(22):7363-72
MexB protein, Pseudomonas aeruginosa
0
*Bacterial Outer Membrane Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
J Bacteriol 1993 Nov;175(22):7363-72
GP-
88, propafenone-
type MDR-
modulator
0
*Phenyl Ethers
*Propanols
Drug Resistance, Multiple.
Bioorg Med Chem Lett 1998 Apr 7;8(7):829-32
ABCG2 protein, human
0
*Neoplasm Proteins
*ATP-Binding Cassette Transporters
Drug Resistance, Multiple.
Biochem Pharmacol. 2005 Jun 23; Proc Natl Acad Sci U S A 1998 Dec 22;95(26):15665-70
Tap protein, Mycobacterium
0
*Bacterial Proteins
*Membrane Transport Proteins
Drug Resistance, Microbial
Drug Resistance, Multiple.
J Bacteriol 1998 Nov;180(22):5836-43
Pmr1 protein, bacteria
0
*Bacterial Proteins
*ATP-Binding Cassette Transporters
Drug Resistance, Multiple.
Appl Environ Microbiol 1998 Oct;64(10):3983-8
multidrug resistance-
associated protein 3
0
*Multidrug Resistance-Associated Proteins
Drug Resistance, Multiple.
FEBS Lett 1998 Aug 14;433(1-2):149-52
ATPGP2 protein, Arabidopsis
0
*ATP-Binding Cassette Transporters
*Arabidopsis Proteins
Drug Resistance, Multiple.
Methods Enzymol 1998;292:162-73
ATPGP1 protein, Arabidopsis
0
*ATP-Binding Cassette Transporters
*Arabidopsis Proteins
Drug Resistance, Multiple.
Methods Enzymol 1998;292:162-73
qacH protein, Staphylococcus saprophyticus
0
*Bacterial Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
FEMS Microbiol Lett 1998 Jan 1;163(1):49-56
hapalosin
159542-04-8
*Lactams
*Lactones
*Depsipeptides
Drug Resistance, Multiple.
J Med Chem 1998 Mar 12;41(6):981-7
MDR1 protein, Filobasidiella neoformans
0
*Fungal Proteins
*ATP-Binding Cassette Transporters
Cryptococcus neoformans
Drug Resistance, Multiple.
Gene 1997 Nov 12;201(1-2):21-9
HIPK3 protein, human
EC 2.7.11.1
*Protein-Serine-Threonine Kinases
*Intracellular Signaling Peptides and Proteins
Drug Resistance, Multiple.
Gene 1997 Oct 24;200(1-2):35-43; J Biol Chem 1998 Oct 2;273(40):25875-9
AadB protein, Acinetobacter sp. SUN
0
*Bacterial Proteins
Drug Resistance, Multiple.
FEMS Microbiol Lett 1997 Aug 15;153(2):321-6
VA 033
0
*Vinca Alkaloids
Drug Resistance, Multiple.
Eur J Pharmacol 1997 May 30;327(2-3):239-46
VX 710
0
*Piperidines
*Pyridines
Drug Resistance, Multiple.
Anticancer Drugs 1997 Feb;8(2):125-40
LmrA protein, Lactococcus lactis
0
*Bacterial Proteins
*Multidrug Resistance-Associated Proteins
Drug Resistance, Multiple.
Proc Natl Acad Sci U S A 1996 Oct 1;93(20):10668-72
QacB protein, Staphylococcus aureus
0
*Bacterial Proteins
*Membrane Transport Proteins
Drug Resistance, Multiple.
Proc Natl Acad Sci U S A 1996 Apr 16;93(8):3630-5
BmrR protein, bacteria
0
*Bacterial Proteins
*Trans-Activators
DNA-Binding Proteins
Drug Resistance, Microbial
Drug Resistance, Multiple.
J Biol Chem 1994 Nov 11;269(45):28506-13
LfrA protein, Mycobacterium smegmatis
0
*Bacterial Proteins
*Antiporters
Drug Resistance, Multiple.
Proc Natl Acad Sci U S A 1996 Jan 9;93(1):362-6
RamA protein, Klebsiella
0
*Bacterial Proteins
Drug Resistance, Multiple.
Microbiology 1995 Aug;141( Pt 8):1909-20
zosuquidar trihydrochloride
0
*Dibenzocycloheptenes
*Quinolines
Drug Resistance, Multiple.
Anticancer Res 1995 May-Jun;15(3):811-4
multidrug resistance protein 3
0
*P-Glycoproteins
Drug Resistance, Multiple.
Hematol Oncol Clin North Am 1995 Apr;9(2):239-49
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